Bromide

Bromide

SCHEMBL27642007

Br.COc1ccc(C(=O)CN2C=CN(c3ccc(C(C)=O)cc3)C2)cc1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 2/20 0.51
LMNA P02545 1/20 0.51
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC5 Q9UQL6 2/20 0.44
MET P08581 1/20 0.43
NPC1 O15118 2/20 0.42
MAPT P10636 2/20 0.41
RAB9A P51151 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3854380 0.86 HTR1A (0.49) ALDH1A1KDM4ELMNAMEN1KMT2A
Bromide SCHEMBL27662427 0.85 MEN1 (0.50) ALDH1A1KDM4ELMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL3851017 0.84 NPC1 (0.41) ALDH1A1LMNAKMT2ANPC1MAPT
Bromide SCHEMBL3853194 0.79 ALDH1A1 (0.56) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL28841407 0.78 ALDH1A1 (0.54) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL27662644 0.77 ALDH1A1 (0.52) ALDH1A1KDM4ELMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL3854520 0.76 ALDH1A1 (0.47) ALDH1A1KDM4ENPC1MAPTRAB9A
SCHEMBL29793985 0.75 GRIN2B (0.49) ALDH1A1KDM4EMEN1KMT2ANPC1
SCHEMBL28953119 0.75 GRIN2B (0.49) ALDH1A1KDM4EMEN1KMT2ANPC1
Hydrochloric Acid SCHEMBL3848508 0.72 GSK3B (0.46) ALDH1A1KDM4EMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100460395-C Aromatic-cyclo and heterocyclo acylmethyl imidazole salts compound and method for preparing same UNIV YUNNAN (CN) 2009-02-11 CN disclosed
CN-1884266-A Aromatic-cyclo and heterocyclo acylmethyl imidazole salts compound and method for preparing same UNIV YUNNAN (CN) 2006-12-27 CN disclosed