SCHEMBL27652123

SCHEMBL27652123

CCOC(=O)C(=O)c1cccc(-c2ccccc2)c1OC(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.43
PDK2 Q15119 1/20 0.41
ALDH1A1 P00352 4/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DHODH Q02127 1/20 0.40
ACHE P22303 2/20 0.39
SCN1A P35498 2/20 0.39
SCN2A Q99250 2/20 0.39
SCN3A Q9NY46 2/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
SCN9A Q15858 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MAPK1 P28482 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
POLB P06746 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11227110 0.81 LMNA (0.57) LMNAALDH1A1MEN1KMT2ADHODH
SCHEMBL27818669 0.80 HNF4A (0.53) LMNAALDH1A1MEN1KMT2ADHODH
SCHEMBL2499425 0.77 CYP11B1 (0.46) LMNAALDH1A1MEN1KMT2AACHE
SCHEMBL1231452 0.77 BCAT2 (0.57) PDK2SCN9A
Hydrochloric Acid SCHEMBL19385254 0.76 BCAT2 (0.56) PDK2SCN9A
SCHEMBL16673206 0.73 PDK2 (0.50) LMNAPDK2ALDH1A1MEN1KMT2A
SCHEMBL16673136 0.72 PDK2 (0.48) LMNAPDK2MEN1KMT2AMAPT
SCHEMBL16672840 0.72 PDK2 (0.48) LMNAPDK2ALDH1A1MEN1KMT2A
SCHEMBL5837400 0.71 TSHR (0.49) LMNAALDH1A1MEN1KMT2AACHE
SCHEMBL28930303 0.70 IGF2BP2 (0.41) LMNAALDH1A1DHODHL3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1805945-A Biaryl substituted thiazoles, oxazoles and imidazoles as sodium channel blockers MERCK & CO INC (US) 2006-07-19 CN disclosed