SCHEMBL27655973

SCHEMBL27655973

CN1CCC(O)(C(C(=O)N2CCN(C(=O)O)CC2)c2cccc(Br)c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 6/20 0.40
CHRM3 P20309 3/20 0.39
HSD17B10 Q99714 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
LMNA P02545 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
SLC6A9 P48067 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27655996 0.90 ALDH1A1 (0.40) CHRM3ALDH1A1TP53LMNANPSR1
SCHEMBL5695482 0.88 ALDH1A1 (0.39) CHRM1CHRM3ALDH1A1TP53LMNA
SCHEMBL3960632 0.88 MTOR (0.41) ALDH1A1TSHRGAA
SCHEMBL27662339 0.88 GRM5 (0.35) CHRM1CHRM3ALDH1A1TP53KDM4E
SCHEMBL27681882 0.86 ALDH1A1 (0.41) ALDH1A1TP53LMNANPSR1TSHR
SCHEMBL3950290 0.86 SLC6A9 (0.39) ALDH1A1TP53SLC6A9KDM4EGAA
SCHEMBL3957138 0.85 BACE1 (0.39) ALDH1A1LMNATSHRMAPK1
SCHEMBL27682053 0.82 KDM4E (0.38) ALDH1A1TP53SLC6A9KDM4EGAA
SCHEMBL3955540 0.82 CHRM3 (0.41) CHRM1CHRM3HSD17B10ALDH1A1TP53
SCHEMBL27662418 0.82 TSHR (0.47) CHRM1CHRM3HSD17B10LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1972920-A Arylalkyl piperazine derivatives for the treatment of conditions ameliorated by monoamine reuptake including vasomotor symptoms WYETH CORP (US) 2007-05-30 CN disclosed
CN-1894226-A Arylalkyl- and cycloalkylalkyl-piperazine derivatives and methods of their use WYETH CORP (US) 2007-01-10 CN disclosed