SCHEMBL27657293

SCHEMBL27657293

NC(=O)N(c1ccc(-c2cccc3snc(N)c23)cc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.62
FLT3 P36888 11/20 0.62
KIT P10721 11/20 0.62
FLT1 P17948 5/20 0.46
CSF1R P07333 4/20 0.46
FLT4 P35916 3/20 0.46
AURKA O14965 2/20 0.46
AURKB Q96GD4 2/20 0.46
ROCK2 O75116 1/20 0.46
FGFR1 P11362 1/20 0.46
RPS6KB1 P23443 1/20 0.46
RPS6KA3 P51812 1/20 0.46
ROCK1 Q13464 1/20 0.46
PLK3 Q9H4B4 1/20 0.46
ABL1 P00519 4/20 0.38
BCR P11274 2/20 0.38
RIPK1 Q13546 1/20 0.37
SLC9A1 P19634 1/20 0.36
FYN P06241 3/20 0.36
TEK Q02763 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27657292 0.85 KDR (0.49) KDRFLT3KITFLT1CSF1R
SCHEMBL27657289 0.83 KDR (0.47) KDRFLT3KITFLT1CSF1R
SCHEMBL4784983 0.80 KDR (0.62) KDRFLT3KITFLT1CSF1R
SCHEMBL27657353 0.80 KDR (0.62) KDRFLT3KITFLT1CSF1R
SCHEMBL419664 0.77 KDR (1.00) KDRFLT3KITFLT1CSF1R
SCHEMBL27657341 0.76 KDR (0.54) KDRFLT3KITFLT1CSF1R
SCHEMBL1703608 0.76 KDR (0.50) KDRFLT3KITFLT1CSF1R
SCHEMBL27636403 0.76 KDR (0.48) KDRFLT3KITFLT1CSF1R
SCHEMBL425369 0.76 KDR (0.49) KDRFLT3KITFLT1CSF1R
SCHEMBL5257214 0.75 KDR (0.51) KDRFLT3KITFLT1CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102417487-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB 2012-04-18 CN claimed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN claimed
CN-102417487-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB 2012-04-18 CN disclosed
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN disclosed
CN-101827584-A Solid dispersion product of N-aryl ureido drugs ABBOTT GMBH & CO KG 2010-09-08 CN disclosed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN disclosed