SCHEMBL27664784

SCHEMBL27664784

CC(C)(C)C(=O)On1ncc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.41
ELANE P08246 2/20 0.40
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
POLB P06746 3/20 0.38
HSD17B10 Q99714 3/20 0.38
TSHR P16473 1/20 0.38
ASAH1 Q13510 2/20 0.37
SLC22A12 Q96S37 1/20 0.37
RAB9A P51151 4/20 0.36
NPC1 O15118 3/20 0.36
KMT2A Q03164 3/20 0.35
RECQL P46063 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TFPI2 P48307 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28251967 0.84 KMO (0.41) KMOELANECYP11B1CYP11B2POLB
SCHEMBL2029059 0.82 KMO (0.44) KMOELANECYP11B1CYP11B2POLB
SCHEMBL3923482 0.82 KMO (0.39) KMOELANECYP11B1CYP11B2POLB
SCHEMBL1162916 0.82 KMO (0.46) KMOELANEPOLBHSD17B10TSHR
SCHEMBL28094503 0.80 CHEK1 (0.43) KMOKMT2AALDH1A1MAPT
SCHEMBL27690302 0.80 HDAC8 (0.39) KMOELANESLC22A12RAB9ANPC1
SCHEMBL27634812 0.80 CHEK1 (0.54) CYP11B1CYP11B2RAB9AKMT2AALDH1A1
SCHEMBL536315 0.79 KMO (0.45) KMOELANEPOLBHSD17B10TSHR
SCHEMBL1854888 0.79 KMO (0.44) KMOELANEPOLBHSD17B10TSHR
SCHEMBL31661024 0.78 CYP11B1 (0.40) KMOELANECYP11B1CYP11B2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102171192-A Indazole compounds ASAHI KASEI PHARMA CORP 2011-08-31 CN claimed
CN-110300751-A Tetra-substituted alkene compounds and their use for treating breast cancer 卫材 R&D 管理有限公司 2019-10-01 CN disclosed
CN-110214137-A As αvThe indazole derivative of integrin antagonists 百时美施贵宝公司 2019-09-06 CN disclosed
CN-104837832-B GDF-8 inhibitors 里格尔药品股份有限公司 2019-04-26 CN disclosed
CN-106458992-B Pyridyl piperidine 默克专利股份公司 2019-03-15 CN disclosed
CN-106458992-A Pyridyl piperidines 默克专利股份公司 2017-02-22 CN disclosed
CN-104755477-A 2-aminopyridine compounds MERCK PATENT GMBH 2015-07-01 CN disclosed
CN-102171191-A Indazole derivative ASAHI KASEI PHARMA CORP 2011-08-31 CN disclosed
CN-102171192-A Indazole compounds ASAHI KASEI PHARMA CORP 2011-08-31 CN disclosed
CN-100558428-C Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2009-11-11 CN disclosed
CN-101489551-A Aminoindazole urea derivatives MERCK PATENT GMBH (DE) 2009-07-22 CN disclosed
CN-101208094-A Pharmacokinetic improved compounds SURFACE LOGIX INC (US) 2008-06-25 CN disclosed
CN-1917921-A Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2007-02-21 CN disclosed