SCHEMBL27665265

SCHEMBL27665265

O=C(O)c1ccc(C(=O)C=Cc2ccc3cc(C(=O)F)ccc3n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 6/20 0.56
CYSLTR2 Q9NS75 2/20 0.53
CYSLTR1 Q9Y271 2/20 0.53
HDAC6 Q9UBN7 4/20 0.50
ALOX5 P09917 1/20 0.45
KDM4E B2RXH2 3/20 0.43
LMNA P02545 2/20 0.43
HDAC8 Q9BY41 3/20 0.41
HDAC3 O15379 2/20 0.41
HDAC4 P56524 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC7 Q8WUI4 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC10 Q969S8 2/20 0.41
HDAC11 Q96DB2 2/20 0.41
HDAC9 Q9UKV0 2/20 0.41
HDAC5 Q9UQL6 2/20 0.41
MAPT P10636 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5090111 0.84 PFKFB3 (0.65) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL5090108 0.84 PFKFB3 (0.65) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL5507715 0.81 PFKFB3 (0.74) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL10275157 0.81 PFKFB3 (0.74) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL5096130 0.80 PFKFB3 (0.52) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL5096126 0.80 PFKFB3 (0.52) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL28289894 0.80 ALOX5 (0.61) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL27684619 0.79 PFKFB3 (0.51) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL28288480 0.77 ALOX5 (0.58) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5
SCHEMBL27985742 0.77 CCR1 (0.41) PFKFB3CYSLTR2CYSLTR1HDAC6ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1964946-A 2-propen-1-ones as HSP 70 inducers TORRENT PHARMACEUTICALS LTD (IN) 2007-05-16 CN disclosed