SCHEMBL27686178

SCHEMBL27686178

NC(=O)c1c(CC(O)N2CCOCC2)c2ncc(Cc3ccc(F)cc3)cc2n(Cc2ccncc2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.39
PDE1B Q01064 3/20 0.34
PDE1A P54750 2/20 0.34
PDE1C Q14123 2/20 0.34
USP2 O75604 5/20 0.33
CASP1 P29466 5/20 0.33
CYP1A2 P05177 5/20 0.33
ALDH1A1 P00352 4/20 0.33
CASP7 P55210 4/20 0.33
HIF1A Q16665 4/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
TSHR P16473 3/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2C9 P11712 3/20 0.33
HPGD P15428 2/20 0.33
CYP2C19 P33261 2/20 0.33
RECQL P46063 1/20 0.33
HSD17B10 Q99714 4/20 0.33
GRM2 Q14416 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28765661 0.87 GRM2 (0.36) ALDH1A1HIF1AMEN1KMT2ATSHR
SCHEMBL27667135 0.87 GRIN2B (0.42) ALDH1A1GRIN2BNTRK1LMNA
SCHEMBL27686172 0.86 GRIN2B (0.40) GRIN2B
SCHEMBL27667098 0.85 GRIN2B (0.39) GRIN2B
SCHEMBL27667115 0.81 OPRM1 (0.35) USP2CASP1ALDH1A1CASP7HIF1A
SCHEMBL27667119 0.80 GRIN2B (0.44) ALDH1A1GRIN2BNTRK1LMNA
SCHEMBL27666972 0.79 NTRK1 (0.36) ALDH1A1HPGDHSD17B10GRM2MAPK1
SCHEMBL27686188 0.79 GRIN1 (0.40) ALDH1A1HPGDRECQLGRM2GRIN2B
SCHEMBL27686159 0.78 CNR2 (0.34) GRM2CNR2CNR1
SCHEMBL27686211 0.76 STAT6 (0.39) PIK3CAUSP2CASP1CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed