SCHEMBL27675186

SCHEMBL27675186

CCc1ccc(NC(=O)n2cc(C(=O)O)c(=O)c3ccccc32)cc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 2/20 0.52
CHRM1 P11229 2/20 0.44
LMNA P02545 2/20 0.43
CREBBP Q92793 2/20 0.42
MAOB P27338 2/20 0.42
EP300 Q09472 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
BLM P54132 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27675185 0.88 CFTR (0.51) CFTRCHRM1LMNACREBBPMAOB
SCHEMBL27693534 0.87 MAOB (0.50) CHRM1LMNACREBBPMAOBEP300
SCHEMBL27693491 0.85 CFTR (0.53) CFTRCHRM1LMNACREBBPMAOB
SCHEMBL27693563 0.85 HSD17B10 (0.41) CFTRCHRM1LMNACREBBPMAOB
SCHEMBL27675310 0.84 CHRM1 (0.54) CFTRCHRM1LMNACREBBPMAOB
SCHEMBL27693546 0.84 LMNA (0.42) CFTRCHRM1LMNACREBBPEP300
SCHEMBL27675123 0.83 CHRM1 (0.42) CHRM1LMNACREBBPMAOBEP300
SCHEMBL27675227 0.82 CFTR (0.48) CFTRCHRM1LMNACREBBPMAOB
SCHEMBL27693645 0.82 CHRM1 (0.54) CHRM1LMNAMEN1KMT2APOLB
SCHEMBL27693487 0.81 LMNA (0.51) CHRM1LMNACREBBPMAOBEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891680-B Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-29 CN disclosed
CN-101935301-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2013-10-16 CN disclosed
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed