SCHEMBL27675205

SCHEMBL27675205

NS(=O)(=O)c1ccccc1NC(=O)n1cc(C(=O)O)c(=O)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.47
USP2 O75604 5/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
CA1 P00915 5/20 0.44
CA2 P00918 5/20 0.44
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
CHRM1 P11229 1/20 0.43
LMNA P02545 5/20 0.43
MEN1 O00255 4/20 0.43
HTT P42858 4/20 0.43
KMT2A Q03164 4/20 0.43
TSHR P16473 3/20 0.43
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
MAPK1 P28482 1/20 0.42
UBE2N P61088 1/20 0.42
HBB P68871 1/20 0.42
TNF P01375 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27675206 0.82 KDM4E (0.48) KDM4ECHRM1LMNAMEN1KMT2A
SCHEMBL27675220 0.82 CA1 (0.49) CA1CA2CA12CA9CHRM1
SCHEMBL27693495 0.81 LMNA (0.49) KDM4ENPC1RAB9ACHRM1LMNA
SCHEMBL28768803 0.81 CNR2 (0.51) KDM4EUSP2NPC1RAB9ALMNA
SCHEMBL27693502 0.81 KDM4E (0.44) KDM4ECHRM1LMNAMEN1KMT2A
SCHEMBL27693559 0.80 KDM4E (0.51) KDM4ERAB9ACHRM1LMNAMEN1
SCHEMBL27693503 0.79 CFTR (0.47) KDM4ECHRM1LMNAALDH1A1HPGD
SCHEMBL27693542 0.79 CNR2 (0.45) KDM4ELMNAKMT2AALDH1A1GAA
SCHEMBL27693487 0.79 LMNA (0.51) KDM4EUSP2CHRM1LMNAMEN1
SCHEMBL28763089 0.78 CFTR (0.48) KDM4ECHRM1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed