SCHEMBL27675271

SCHEMBL27675271

O=C(O)c1cn(C(=O)Nc2ccccc2N2CCCCC2)c2ccccc2c1=O

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 7/20 0.48
L3MBTL1 Q9Y468 4/20 0.48
MAPT P10636 2/20 0.48
TSHR P16473 3/20 0.46
ATM Q13315 2/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
USP2 O75604 1/20 0.46
GLA P06280 1/20 0.46
HTT P42858 1/20 0.46
KCNQ2 O43526 4/20 0.46
KMT2A Q03164 3/20 0.46
GAA P10253 3/20 0.46
PKM P14618 1/20 0.46
LMNA P02545 3/20 0.45
MEN1 O00255 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPK1 P28482 1/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27693573 0.89 CASP3 (0.53) NPSR1L3MBTL1MAPTALDH1A1USP2
SCHEMBL27675288 0.87 TSHR (0.53) NPSR1MAPTTSHRALDH1A1KDM4E
SCHEMBL28768803 0.79 CNR2 (0.51) MAPTTSHRALDH1A1KDM4EUSP2
SCHEMBL27693495 0.79 LMNA (0.49) MAPTALDH1A1KDM4EKMT2ALMNA
SCHEMBL27675206 0.78 KDM4E (0.48) MAPTALDH1A1KDM4EKMT2AGAA
SCHEMBL27693559 0.78 KDM4E (0.51) L3MBTL1MAPTALDH1A1KDM4EHTT
SCHEMBL27693542 0.77 CNR2 (0.45) MAPTALDH1A1KDM4EKMT2AGAA
SCHEMBL27693503 0.77 CFTR (0.47) ALDH1A1KDM4ELMNAPOLB
SCHEMBL27693487 0.77 LMNA (0.51) TSHRALDH1A1KDM4EUSP2HTT
SCHEMBL28763089 0.76 CFTR (0.48) ALDH1A1KDM4EKMT2ALMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed