SCHEMBL27680901

SCHEMBL27680901

O=[N+]([O-])c1cccc(-c2cc(C3CNCCO3)nc(-c3cccc(CO)c3)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.38
IDO1 P14902 1/20 0.38
ALDH1A1 P00352 6/20 0.38
MAPT P10636 5/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
POLB P06746 1/20 0.38
MTOR P42345 4/20 0.37
MAPK1 P28482 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
PIK3CA P42336 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PIK3CG P48736 1/20 0.35
THRB P10828 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27685978 1.00 VCP (0.38) VCPIDO1ALDH1A1MAPTMEN1
SCHEMBL27686021 0.84 ALDH1A1 (0.37) VCPIDO1ALDH1A1MAPTMEN1
SCHEMBL27700074 0.84 KDM4E (0.43) ALDH1A1MAPTMEN1KMT2AMTOR
SCHEMBL27705039 0.84 KDM4E (0.43) ALDH1A1MAPTMEN1KMT2AMTOR
SCHEMBL27682784 0.83 NPC1 (0.41) IDO1ALDH1A1MAPTMEN1KMT2A
SCHEMBL27685979 0.82 CYP1A2 (0.40) IDO1ALDH1A1MAPTMEN1KMT2A
SCHEMBL27680902 0.82 CYP1A2 (0.40) IDO1ALDH1A1MAPTMEN1KMT2A
SCHEMBL27700082 0.82 MEN1 (0.40) ALDH1A1MAPTMEN1KMT2AMTOR
SCHEMBL27680908 0.82 IDO1 (0.40) VCPIDO1ALDH1A1MAPTMEN1
SCHEMBL27680857 0.81 SLC6A3 (0.42) MTORPIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101010317-A 2, 4,6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer ASTRAZENECA AB (SE) 2007-08-01 CN disclosed