SCHEMBL27680906

SCHEMBL27680906

Nc1cccc(-c2cc(C3CNCCO3)ncn2)c1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRKACA P17612 1/20 0.43
PRKACG P22612 1/20 0.43
PRKACB P22694 1/20 0.43
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27700096 0.87 PRKACA (0.42) PRKACAPRKACGPRKACBDRD2DRD3
SCHEMBL27700080 0.82 PRKACA (0.41) PRKACAPRKACGPRKACBDRD2DRD3
SCHEMBL28900236 0.77 DRD2 (0.46) DRD2DRD3HTR1A
SCHEMBL27682789 0.76 PRKACA (0.43) PRKACAPRKACGPRKACBDRD2DRD3
SCHEMBL27700074 0.76 KDM4E (0.43) PRKACAPRKACGPRKACBDRD2DRD3
SCHEMBL27705039 0.76 KDM4E (0.43) PRKACAPRKACGPRKACBDRD2DRD3
SCHEMBL6389994 0.74 DRD2 (0.68) PRKACAPRKACGPRKACBDRD2DRD3
SCHEMBL18399274 0.73 DRD2 (0.43) DRD2DRD3HTR1A
SCHEMBL18399078 0.73 SLC6A3 (0.46)
SCHEMBL27482516 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101010317-A 2, 4,6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer ASTRAZENECA AB (SE) 2007-08-01 CN disclosed