SCHEMBL27680951

SCHEMBL27680951

CCCCn1c(C=O)cnc1C1CC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 7/20 0.35
PDE1A P54750 6/20 0.35
PDE1B Q01064 6/20 0.35
PARP1 P09874 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE4D Q08499 6/20 0.32
PDE6A P16499 1/20 0.32
PDE6B P35913 1/20 0.32
PDE4A P27815 4/20 0.31
ADORA2A P29274 4/20 0.31
PDE4B Q07343 4/20 0.31
PDE4C Q08493 4/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADORA2B P29275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27660999 0.76 ALDH1A1 (0.40) MEN1KMT2APDE4DPDE4AADORA2A
SCHEMBL4036563 0.76 PDE1B (0.35) PDE1CPDE1APDE1BTDP1
SCHEMBL4031313 0.71 PDE1B (0.35) PDE1CPDE1APDE1BADORA2AADORA2B
SCHEMBL27493137 0.70 ADORA2A (0.36) PDE1CPDE1APDE1BADORA2ATDP1
SCHEMBL650017 0.70 TSHR (0.56) PDE4BTDP1L3MBTL1ADORA2B
SCHEMBL4034699 0.69 CDK2 (0.36)
SCHEMBL21435153 0.66 KEAP1 (0.32)
SCHEMBL9454065 0.65
SCHEMBL14557025 0.64 KMT2A (0.35) PDE1CPDE1APDE1BMEN1KMT2A
SCHEMBL7398877 0.64 AGTR1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1930144-A 3-'4-heterocyclyl -1,2,3,-triazol-1-yl!-n-aryl-benzamides as inhibitors of the cytokines production for the treatment of chronic inflammatory diseases BOEHRINGER INGELHEIM PHARMA (US) 2007-03-14 CN disclosed