SCHEMBL27684231

SCHEMBL27684231

Nc1cncnc1Oc1ccc(I)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.35
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
ICAM1 P05362 1/20 0.33
SELE P16581 1/20 0.33
TRPA1 O75762 2/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
APEX1 P27695 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
NSD2 O96028 1/20 0.31
NSD3 Q9BZ95 1/20 0.31
RET P07949 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAP3K8 P41279 1/20 0.31
MEN1 O00255 1/20 0.31
APAF1 O14727 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27664617 0.82 TRPA1 (0.46) TRPA1CYP2C9TSHRALDH1A1MEN1
SCHEMBL20406319 0.79 APP (0.35) APPLMNAICAM1SELETRPA1
SCHEMBL10033148 0.79 RAB9A (0.51) LMNAMAPTICAM1SELECYP2C9
SCHEMBL1803089 0.74 MEN1 (0.43) APPMAPTALDH1A1MEN1APAF1
SCHEMBL28803764 0.73 TRPA1 (0.33) TRPA1
SCHEMBL20406329 0.69 CYP2C9 (0.43) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL5735866 0.67
SCHEMBL31008552 0.67
SCHEMBL20406283 0.66 KDM4E (0.49) LMNAMAPTSMN1; SMN2ALDH1A1MEN1
SCHEMBL20406284 0.66 TRPA1 (0.31) LMNATRPA1CYP2C9TSHRAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1993362-B Fused Heterocyclic Compounds TAKEDA PHARMACEUTICAL 2010-12-15 CN disclosed
CN-1993362-A Fused Heterocyclic Compounds TAKEDA PHARMACEUTICAL (JP) 2007-07-04 CN disclosed