SCHEMBL27685083

SCHEMBL27685083

CC(Br)c1cccc(SC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
P2RX7 Q99572 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CETP P11597 2/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
CASR P41180 1/20 0.32
RXFP1 Q9HBX9 2/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KCNH2 Q12809 1/20 0.31
TRPV1 Q8NER1 3/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12610671 0.85 ALDH1A1 (0.41) KDM4EALDH1A1TDP1SMN1; SMN2CETP
SCHEMBL4550392 0.82 KDM4E (0.38) KDM4EALDH1A1TDP1SMN1; SMN2CETP
Hydrochloric Acid SCHEMBL2717881 0.81 KDM4E (0.37) KDM4EALDH1A1TDP1SMN1; SMN2CETP
SCHEMBL24781619 0.79 HDAC4 (0.45) KDM4EALDH1A1TDP1SMN1; SMN2CETP
SCHEMBL27797879 0.78 MAPT (0.39) KDM4EALDH1A1SMN1; SMN2CETPLMNA
SCHEMBL27797880 0.78 LMNA (0.33) KDM4EALDH1A1TDP1SMN1; SMN2CETP
SCHEMBL27606147 0.78 RXFP1 (0.38) KDM4EALDH1A1TDP1SMN1; SMN2CETP
SCHEMBL1721080 0.77 KDM4E (0.48) KDM4EALDH1A1TDP1SMN1; SMN2LMNA
SCHEMBL28041626 0.77 CYP3A4 (0.41) SMN1; SMN2MAPTMAPK1KCNH2POLB
SCHEMBL11166250 0.76 ESR1 (0.36) KDM4EALDH1A1TDP1SMN1; SMN2CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101048382-B Novel indole or benzimidazole derivatives HOFFMANN LA ROCHE 2010-05-05 CN disclosed
CN-101048382-A Novel Indole or Benzimidazole Derivatives HOFFMANN LA ROCHE (CH) 2007-10-03 CN disclosed