SCHEMBL27686161

SCHEMBL27686161

NC(=O)c1c(CC(O)CO)c2ncc(Cc3ccc(F)cc3)cc2n(CC2CC2)c1=O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.33
GRM2 Q14416 9/20 0.33
SCN9A Q15858 3/20 0.33
LMNA P02545 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
KCNH2 Q12809 1/20 0.31
CYP3A4 P08684 1/20 0.30
NPC1 O15118 1/20 0.30
ROCK2 O75116 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27686289 0.92 LMNA (0.33) GRM2LMNARXFP1CYP3A4NPC1
SCHEMBL6061367 0.90 GRM2 (0.35) GRM2LMNARXFP1KCNH2CYP3A4
SCHEMBL27667069 0.87 FEN1 (0.34) GRM2SCN9A
SCHEMBL27667167 0.86 TRPC5 (0.37) GRM2SCN9AKCNH2
SCHEMBL27686095 0.84 GRIN2B (0.40)
SCHEMBL27686146 0.84 CNR2 (0.33) GRM2SCN9A
SCHEMBL27686312 0.83 GRIN1 (0.37) GRM2LMNA
SCHEMBL27667205 0.83 GRM2 (0.39) TRPV1GRM2SCN9AKCNH2
SCHEMBL27686092 0.83 GRM2 (0.39) TRPV1GRM2SCN9AKCNH2CYP3A4
SCHEMBL27686081 0.82 LMNA (0.35) GRM2LMNARXFP1KCNH2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed