SCHEMBL2768641

SCHEMBL2768641

CCN(C(=O)OC(C)(C)C)c1nc2[nH]c(-c3cccc(Cl)n3)cc2c2[nH]cnc12

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 18/20 0.34
PIM1 P11309 2/20 0.33
PIM2 Q9P1W9 2/20 0.33
CHUK O15111 1/20 0.32
RET P07949 1/20 0.32
CYP2C9 P11712 1/20 0.32
EPHA1 P21709 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
EPHB1 P54762 1/20 0.32
PTK6 Q13882 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2766679 0.89 IKBKB (0.46) IKBKB
SCHEMBL2766834 0.86 IKBKB (0.41) IKBKBCHUKRETCYP2C9EPHA1
SCHEMBL3037384 0.85 IKBKB (0.48) IKBKB
SCHEMBL2767729 0.80 CHUK (0.31) IKBKBPIM1PIM2CHUK
SCHEMBL2767778 0.79 MEN1 (0.33)
SCHEMBL2767620 0.78 EGFR (0.36)
SCHEMBL3041370 0.77 L3MBTL1 (0.36) IKBKBCHUK
SCHEMBL2767746 0.77 TBK1 (0.33)
SCHEMBL2767074 0.76 IKBKB (0.30) IKBKBCHUK
SCHEMBL2768532 0.76 NLRP3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881967-B1 SUBSTITUTED BENZO(D)ISOXAZOL-3-YL AMINE COMPOUNDS AS ANALGESICS GRUENENTHAL GMBH (DE) 2010-04-28 EP claimed
EP-1881967-B1 SUBSTITUTED BENZO(D)ISOXAZOL-3-YL AMINE COMPOUNDS AS ANALGESICS GRUENENTHAL GMBH (DE) 2010-04-28 EP disclosed