SCHEMBL27691593

SCHEMBL27691593

O=c1[nH]c(=O)n(COCc2ccccc2)c(Cc2ccccc2)c1I

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
UPP1 Q16831 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TK1 P04183 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
TSHR P16473 1/20 0.37
HPGD P15428 2/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
DAO P14920 4/20 0.36
USP2 O75604 1/20 0.35
MAPK1 P28482 1/20 0.35
LMNA P02545 1/20 0.35
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27691588 0.88 ALDH1A1 (0.45) ALDH1A1UPP1CYP2C9CYP2C19TSHR
SCHEMBL27691590 0.84 ALDH1A1 (0.70) ALDH1A1UPP1CYP2C9CYP2C19TK1
SCHEMBL27691591 0.82 ALDH1A1 (0.56) ALDH1A1UPP1CYP2C9CYP2C19TK1
SCHEMBL27691587 0.81 HPGD (0.50) ALDH1A1SMN1; SMN2TSHRHPGDKDM4E
SCHEMBL30601622 0.81 ALDH1A1 (0.55) ALDH1A1UPP1CYP2C9CYP2C19TK1
SCHEMBL6719602 0.73 ALDH1A1 (0.75) ALDH1A1UPP1CYP2C9CYP2C19TK1
SCHEMBL6723373 0.73 ALDH1A1 (0.59) ALDH1A1CYP2C9CYP2C19TK1SMN1; SMN2
SCHEMBL5383431 0.72 ALDH1A1 (0.51) ALDH1A1UPP1CYP2C9CYP2C19TK1
SCHEMBL598947 0.72 ALDH1A1 (0.45) ALDH1A1UPP1CYP2C9CYP2C19SMN1; SMN2
SCHEMBL27711771 0.72 ALDH1A1 (0.57) ALDH1A1UPP1CYP2C9CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102838549-A New class of 1,5,6-substituted pyrimidine derivatives with anti-HIV virus effects UNIV BEIJING 2012-12-26 CN claimed
CN-101016265-A Preparation of HIV-1 reverse transcriptase inhibitor and application thereof UNIV CAPITAL MEDICAL SCIENCES (CN) 2007-08-15 CN claimed
CN-102838549-A New class of 1,5,6-substituted pyrimidine derivatives with anti-HIV virus effects UNIV BEIJING 2012-12-26 CN disclosed
CN-101016265-A Preparation of HIV-1 reverse transcriptase inhibitor and application thereof UNIV CAPITAL MEDICAL SCIENCES (CN) 2007-08-15 CN disclosed