SCHEMBL6723373

SCHEMBL6723373

O=c1[nH]c(=O)n(COCc2ccccc2)c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.59
P2RX4 Q99571 1/20 0.44
DAO P14920 1/20 0.43
PARP1 P09874 5/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
TK1 P04183 1/20 0.42
CYP19A1 P11511 1/20 0.41
KDM4E B2RXH2 2/20 0.41
CYP1A2 P05177 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PGR P06401 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 2/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30728403 0.81 CYP19A1 (0.57) ALDH1A1P2RX4CYP2C19CYP19A1KDM4E
SCHEMBL6719104 0.78 NPC1 (0.53) ALDH1A1DAOPARP1CYP2C9KDM4E
SCHEMBL2980047 0.78 ALDH1A1 (0.54) ALDH1A1DAOPARP1CYP2C9CYP2C19
SCHEMBL6731313 0.78 ALDH1A1 (0.50) ALDH1A1P2RX4DAOPARP1KDM4E
SCHEMBL6719602 0.77 ALDH1A1 (0.75) ALDH1A1DAOCYP2C9CYP2C19TK1
SCHEMBL6027805 0.74 CYP1A2 (0.64) ALDH1A1DAOPARP1KDM4ECYP1A2
SCHEMBL8377270 0.74 KDM4E (0.64) ALDH1A1PARP1KDM4E
SCHEMBL27691590 0.73 ALDH1A1 (0.70) ALDH1A1DAOCYP2C9CYP2C19TK1
SCHEMBL27691593 0.73 ALDH1A1 (0.55) ALDH1A1DAOCYP2C9CYP2C19TK1
SCHEMBL9394061 0.73 ALDH1A1 (0.51) ALDH1A1CYP2C9CYP2C19TK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6673804-B1 PREVENTING OR TREATING ARTHRITIS (PARTICULARLY OSTEOARTHRITIS) OR INHIBITING METASTASIS, INVASION OR GROWTH OF CANCER (PARTICULARLY BREAST CANCER) SANKYO COMPANY, LIMITED (JP) 2004-01-06 US disclosed
EP-1069110-A1 SULFONAMIDE DERIVATIVES Sankyo Company Limited (JP) 2001-01-17 EP disclosed