SCHEMBL27694757

SCHEMBL27694757

O=C(Nc1cccnc1)c1cc(-c2ccc(F)cc2)n(-c2ccccc2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.57
PTGS1 P23219 1/20 0.56
PTGS2 P35354 1/20 0.56
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
MALT1 Q9UDY8 2/20 0.54
MAPK9 P45984 1/20 0.53
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
ATM Q13315 1/20 0.53
MARS1 P56192 2/20 0.52
CACNA1G O43497 2/20 0.50
CACNA1H O95180 2/20 0.50
NAMPT P43490 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NPC1 O15118 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
RAB9A P51151 1/20 0.49
RPA1 P27694 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27694750 0.87 TDP1 (0.54) TDP1PTGS1PTGS2MEN1KMT2A
SCHEMBL5483244 0.85 TAAR1 (0.50) TDP1PTGS1PTGS2MEN1KMT2A
SCHEMBL27885071 0.81 MAPK9 (0.58) PTGS1PTGS2MEN1KMT2AMALT1
SCHEMBL9207571 0.80 PTGS2 (0.58) PTGS1PTGS2MEN1KMT2AMALT1
SCHEMBL9206453 0.79 PTGS2 (0.67) PTGS1PTGS2MEN1KMT2AMALT1
SCHEMBL6350064 0.79 PTGS2 (0.82) PTGS1PTGS2MAPK9
SCHEMBL27714729 0.78 KMT2A (0.89) MEN1KMT2AATMMARS1L3MBTL1
SCHEMBL27714718 0.77 KMT2A (0.57) PTGS1PTGS2MEN1KMT2AMALT1
SCHEMBL27694758 0.76 CACNA1G (0.84) PTGS2MEN1KMT2AMALT1ATM
SCHEMBL27694888 0.75 KMT2A (0.71) PTGS2MEN1KMT2AMALT1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101062916-A Three-substituted 1H-pyrromonazole compound, preparation method, medicament composition and pharmacy use thereof POISON MED INST PLA MED ACAD (CN) 2007-10-31 CN claimed
CN-101062916-B Three-substituted 1H-pyrromonazole compound, preparation method, medicament composition and pharmacy use thereof INST PHARM & TOXICOLOGY AMMS 2012-12-26 CN disclosed
CN-101062916-A Three-substituted 1H-pyrromonazole compound, preparation method, medicament composition and pharmacy use thereof POISON MED INST PLA MED ACAD (CN) 2007-10-31 CN disclosed