SCHEMBL27698702

SCHEMBL27698702

CC(C)(C)C(=O)ON1CCN(c2ncc(Br)s2)CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 8/20 0.41
HDAC4 P56524 8/20 0.41
HDAC1 Q13547 8/20 0.41
HDAC7 Q8WUI4 8/20 0.41
HDAC2 Q92769 8/20 0.41
HDAC10 Q969S8 8/20 0.41
HDAC11 Q96DB2 8/20 0.41
HDAC8 Q9BY41 8/20 0.41
HDAC6 Q9UBN7 8/20 0.41
HDAC9 Q9UKV0 8/20 0.41
HDAC5 Q9UQL6 8/20 0.41
TDP1 Q9NUW8 1/20 0.38
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 2/20 0.34
MLYCD O95822 3/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27718997 0.83 HDAC3 (0.36) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL27718993 0.83 MLYCD (0.44) MLYCD
SCHEMBL27719002 0.82 MLYCD (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL27556099 0.82 HRH3 (0.37) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL27698692 0.80 HDAC3 (0.34) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28771983 0.80 HDAC3 (0.34) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28781197 0.79 MLYCD (0.33) TP53MLYCD
SCHEMBL1199336 0.78 GPR119 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL27808994 0.77 RAB9A (0.38) NPC1RAB9ATP53ALDH1A1MAPT
SCHEMBL27718995 0.77 CCNE2 (0.35) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903320-A Nitrogen-containing heterocylic compound or salt thereof FUJIFILM CORP 2015-09-09 CN disclosed
CN-101137363-B [4- (heteroaryl) piperazin-1-yl ] - (2, 5-substituted-phenyl) methanone derivatives as glycine transporter 1(GlyT-1) inhibitors for the treatment of neurological and neuropsychiatric disorders HOFFMANN LA ROCHE 2010-09-15 CN disclosed
CN-101415674-A Pyrrolidine derivatives as ERK inhibitors SCHERING CORP (US) 2009-04-22 CN disclosed
CN-101137363-A [ 4- (heteroaryl) piperazin-1-yl ] - (2, 5-substituted-phenyl) methanone derivatives as glycine transporter 1 (GlyT-1) inhibitors for the treatment of neurological and neuropsychiatric disorders HOFFMANN LA ROCHE (CH) 2008-03-05 CN disclosed