SCHEMBL27699323

SCHEMBL27699323

CCOC(=S)Sc1ccc(F)c(CN)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
HDAC9 Q9UKV0 1/20 0.30
HDAC5 Q9UQL6 1/20 0.30
HPGD P15428 1/20 0.30
ALOX15 P16050 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27719945 0.83 SMN1; SMN2 (0.34) ALDH1A1KDM4EMAPTPKMSMN1; SMN2
SCHEMBL595607 0.82 ALDH1A1 (0.34) ALDH1A1KDM4EMAPTPKMSMN1; SMN2
SCHEMBL6974279 0.79 DHODH (0.34) ALDH1A1KDM4EMAPTPKMSMN1; SMN2
SCHEMBL1632856 0.77 MAPT (0.35) ALDH1A1KDM4EMAPTPKMSMN1; SMN2
SCHEMBL595968 0.75 HTT (0.40) ALDH1A1KDM4ESMN1; SMN2HDAC3HDAC4
SCHEMBL10593979 0.75 MAPT (0.40) ALDH1A1KDM4EMAPTSMN1; SMN2TDP1
SCHEMBL15956317 0.74 ALDH1A1 (0.39) ALDH1A1TDP1HDAC3HDAC4HDAC1
SCHEMBL596880 0.72 ALDH1A1 (0.35) ALDH1A1KDM4EMAPTPKMSMN1; SMN2
SCHEMBL27858862 0.70 LOXL2 (0.36) MAPT
SCHEMBL596873 0.70 MCL1 (0.36) ALDH1A1KDM4EMAPTPKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101163678-B Pyridylmethylsulfone derivative DAIICHI SANKYO CO LTD 2012-01-04 CN disclosed
CN-101163678-A Pyridylmethylsulfone derivative DAIICHI SANKYO CO LTD (JP) 2008-04-16 CN disclosed