SCHEMBL27700950

SCHEMBL27700950

Cc1c(NC(F)(F)F)ncnc1-c1ccc2cccnc2n1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 6/20 0.39
MIF P14174 1/20 0.34
ALDH1A1 P00352 1/20 0.33
SUCNR1 Q9BXA5 6/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPK3 P27361 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6033545 0.82 TRPV1 (0.61) TRPV1
SCHEMBL6033649 0.79 TRPV1 (0.54) TRPV1MAPK3
SCHEMBL6033641 0.75 TRPV1 (0.54) TRPV1MAPK3
SCHEMBL27681512 0.74 CCR1 (0.36) ALDH1A1KDM4ELMNA
SCHEMBL27681517 0.73 TRPV1 (0.42) TRPV1MIFALDH1A1SUCNR1KDM4E
SCHEMBL5801087 0.72 TRPV1 (0.56) TRPV1
SCHEMBL5809097 0.71 TRPV1 (0.57) TRPV1
SCHEMBL1089189 0.67 ALDH1A1 (0.55) MIFALDH1A1KDM4EMEN1LMNA
SCHEMBL27700674 0.65 MTOR (0.37) TRPV1
SCHEMBL18806846 0.65 ALDH1A1 (0.48) MIFALDH1A1SUCNR1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101035780-A Substituted nitrogen-containing six-membered amino-heterocycles as vanilloid-1 receptor antagonists for treating pain MERCK SHARP & DOHME (GB) 2007-09-12 CN claimed
CN-101035780-A Substituted nitrogen-containing six-membered amino-heterocycles as vanilloid-1 receptor antagonists for treating pain MERCK SHARP & DOHME (GB) 2007-09-12 CN disclosed