SCHEMBL27702018

SCHEMBL27702018

N#Cc1cc(F)cc(C#Cc2ccc(CN)cc2)c1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.58
GRM5 P41594 1/20 0.42
FFAR1 O14842 1/20 0.42
ASIC3 Q9UHC3 1/20 0.41
PLAU P00749 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27722556 0.86 LOXL2 (0.44) LOXL2GRM5FFAR1ASIC3
SCHEMBL4460258 0.84 GRM5 (0.50) GRM5
SCHEMBL4457929 0.80 GRM5 (0.56) GRM5
SCHEMBL319482 0.78 LOXL2 (0.48) LOXL2GRM5
SCHEMBL30335660 0.78 LOXL2 (0.48) LOXL2GRM5
SCHEMBL11782098 0.78 LOXL2 (0.73) LOXL2FFAR1ASIC3PLAU
SCHEMBL4454176 0.77 ALDH1A1 (0.54) GRM5
SCHEMBL2758337 0.77 TSHR (0.50) GRM5
SCHEMBL4454587 0.77 HAO1 (0.48) GRM5
Water SCHEMBL5709165 0.75 LOXL2 (1.00) LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101163667-A Phenylacetylene compounds MERCK & CO INC (US) 2008-04-16 CN disclosed