SCHEMBL2770591

SCHEMBL2770591

NC(=O)c1ccc(F)c(F)c1C1CC1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.42
CES1 P23141 4/20 0.42
DGAT1 O75907 1/20 0.41
PARP10 Q53GL7 2/20 0.39
PARP15 Q460N3 1/20 0.39
MAP2K2 P36507 1/20 0.39
MAP2K1 Q02750 1/20 0.39
HTR1A P08908 1/20 0.39
SCN9A Q15858 2/20 0.37
PARP1 P09874 2/20 0.36
ROCK2 O75116 1/20 0.36
MAPK1 P28482 1/20 0.34
EPHX2 P34913 3/20 0.33
HTR5A P47898 1/20 0.33
BCHE P06276 1/20 0.33
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6466321 0.94 ROCK2 (0.44) CES2CES1DGAT1PARP10PARP15
SCHEMBL6466316 0.94 ROCK2 (0.44) CES2CES1DGAT1PARP10PARP15
SCHEMBL5670138 0.89 PARP10 (0.39) CES2CES1DGAT1PARP10PARP15
SCHEMBL4191551 0.86 HTR1A (0.42) CES2CES1DGAT1PARP10PARP15
SCHEMBL10449035 0.82 MAPT (0.38) DGAT1PARP10PARP15PARP1MAPK1
SCHEMBL28182486 0.79 DGAT1 (0.36) CES2CES1DGAT1PARP10PARP15
SCHEMBL31069789 0.79 PARP10 (0.41) PARP10PARP15SCN9AMAPK1
SCHEMBL1116601 0.79 ABCB1 (0.41) CES2CES1PARP1BCHE
SCHEMBL27652684 0.78 ROCK2 (0.43) DGAT1PARP10PARP15HTR1ASCN9A
SCHEMBL813186 0.75 MEN1 (0.46) PARP10PARP15PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111626-A2 POLY (ADP-RIBOSE) POLYMERASE (PARP) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed