SCHEMBL27707635

SCHEMBL27707635

CC=Cc1cc(F)ccc1Br

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
F2RL1 P55085 2/20 0.40
NFE2L2 Q16236 8/20 0.38
HRH4 Q9H3N8 1/20 0.37
AMY1A P0DUB6 1/20 0.36
RELA Q04206 1/20 0.35
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
BACE1 P56817 1/20 0.33
PKM P14618 1/20 0.33
HMGCR P04035 1/20 0.32
CYP3A4 P08684 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22001870 1.00 F2RL1 (0.40) F2RL1NFE2L2HRH4AMY1ARELA
SCHEMBL27563320 0.83 AMY1A (0.38) NFE2L2AMY1ARELAFFAR1FFAR4
SCHEMBL10245246 0.79 ESR1 (0.36) NFE2L2AMY1ARELAFFAR1FFAR4
SCHEMBL876257 0.79 NFE2L2 (0.39) NFE2L2AMY1ARELAPKM
SCHEMBL15093161 0.79 NFE2L2 (0.39) NFE2L2AMY1ARELAPKM
SCHEMBL16951286 0.78 NFE2L2 (0.61) F2RL1NFE2L2HRH4PTGS1PTGS2
SCHEMBL14541331 0.78 NFE2L2 (0.61) F2RL1NFE2L2HRH4PTGS1PTGS2
SCHEMBL16308833 0.77 ALOX5 (0.35) BACE1HMGCRCYP3A4PTGS1PTGS2
SCHEMBL15792855 0.77 ALOX5 (0.35) BACE1HMGCRCYP3A4PTGS1PTGS2
SCHEMBL19337428 0.77 F2RL1 (0.41) F2RL1NFE2L2HRH4FFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101048414-B Fused tricyclic derivatives for the treatment of psychotic disorders GLAXO GROUP LTD 2011-09-07 CN disclosed
CN-101048414-A Fused tricyclic derivatives for the treatment of psychotic disorders GLAXO GROUP LTD (GB) 2007-10-03 CN disclosed