SCHEMBL27709059

SCHEMBL27709059

C[C@@H](CNC(=O)c1cc2cc(Cl)ccc2[nH]1)CC(=N)C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.55
HRH3 Q9Y5N1 1/20 0.55
PYGL P06737 12/20 0.54
NHERF1 O14745 1/20 0.52
CNR1 P21554 1/20 0.49
F7 P08709 1/20 0.49
F3 P13726 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27709042 0.91 ALOX15 (0.60) HRH4HRH3PYGL
SCHEMBL6350243 0.79 PYGL (0.62) HRH4HRH3PYGLNHERF1F7
SCHEMBL5869858 0.77 PYGL (0.56) HRH4HRH3PYGLNHERF1
SCHEMBL5869825 0.77 PYGL (0.56) HRH4HRH3PYGLNHERF1
SCHEMBL5869836 0.77 PYGL (0.56) HRH4HRH3PYGLNHERF1
SCHEMBL27709050 0.76 MEN1 (0.48)
SCHEMBL27729464 0.76 OPRM1 (0.49)
SCHEMBL13753365 0.76 ALOX15 (0.79) HRH4HRH3PYGLNHERF1CNR1
SCHEMBL2410978 0.76 HDAC3 (0.56) HRH4HRH3PYGLNHERF1CNR1
SCHEMBL28757959 0.75 PYGL (0.50) HRH4HRH3PYGLNHERF1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101208334-B Novel cyclic amines HOFFMANN LA ROCHE 2012-06-13 CN disclosed
CN-101208334-A Novel cyclic amines HOFFMANN LA ROCHE (CH) 2008-06-25 CN disclosed