SCHEMBL27710141

SCHEMBL27710141

Cc1c(C(=O)O)ccc(-c2cccc3[nH]ccc23)c1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 1/20 0.45
BTK Q06187 5/20 0.41
PIK3CD O00329 1/20 0.40
MAPK14 Q16539 2/20 0.40
AHR P35869 1/20 0.39
DHFR P00374 1/20 0.38
ASH1L Q9NR48 1/20 0.38
HPGDS O60760 2/20 0.38
MCL1 Q07820 1/20 0.38
AURKA O14965 1/20 0.38
TPX2 Q9ULW0 1/20 0.38
PDE10A Q9Y233 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27710092 0.83 PDE10A (0.49) PDE10A
SCHEMBL1570156 0.79 FTO (0.56) FTOPIK3CDMAPK14ASH1LHPGDS
SCHEMBL27690173 0.78 METAP2 (0.49) AURKA
SCHEMBL14559813 0.77 P2RX7 (0.50) AHRMCL1AURKATPX2
SCHEMBL27487899 0.77 KDM4E (0.58) MCL1PDE10A
SCHEMBL27624407 0.74 MYC (0.50) DHFRMCL1
SCHEMBL28207084 0.74 MYC (0.53)
SCHEMBL27844241 0.74 NAPRT (0.42) AURKATPX2
SCHEMBL29684913 0.73 NAPRT (0.52) FTOMAPK14AHR
SCHEMBL40257 0.73 NAPRT (0.52) FTOMAPK14AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101119969-A Aryl and heteroaryl substituted tetrahydroisoquinolines and their use to block reuptake of norepinephrine, dopamine, and serotonin AMR TECHNOLOGY INC (US) 2008-02-06 CN claimed
CN-103880827-A Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin ALBANY MOLECULAR RES INC 2014-06-25 CN disclosed
CN-101119969-A Aryl and heteroaryl substituted tetrahydroisoquinolines and their use to block reuptake of norepinephrine, dopamine, and serotonin AMR TECHNOLOGY INC (US) 2008-02-06 CN disclosed