Quinoline

Quinoline

SCHEMBL27713201

Fc1ccc2cc[nH]c2c1.c1ccc2ncccc2c1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 5/20 0.62
ALDH1A1 P00352 4/20 0.50
METAP2 P50579 1/20 0.43
METAP1 P53582 1/20 0.43
CBFB Q13951 1/20 0.43
NR4A2 P43354 1/20 0.42
TRPA1 O75762 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
ITGB2 P05107 1/20 0.42
ICAM1 P05362 1/20 0.42
ITGAL P20701 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
ADK P55263 1/20 0.42
AXL P30530 1/20 0.41
NUDT1 P36639 1/20 0.41
CYP1A2 P05177 2/20 0.39
MEN1 O00255 1/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27717739 0.88 AHR (0.62) AHRALDH1A1METAP2METAP1CBFB
Quinoline SCHEMBL28073739 0.82 ALDH1A1 (0.63) AHRALDH1A1METAP2METAP1NR4A2
Quinoline SCHEMBL843861 0.82 ALDH1A1 (0.63) AHRALDH1A1METAP2METAP1NR4A2
Quinoline SCHEMBL28292512 0.82 ALDH1A1 (0.63) AHRALDH1A1METAP2METAP1NR4A2
Quinoline SCHEMBL28816675 0.82 ALDH1A1 (0.63) AHRALDH1A1METAP2METAP1NR4A2
Quinoline SCHEMBL28212903 0.82 AHR (0.54) AHRALDH1A1METAP2METAP1CBFB
Quinoline SCHEMBL28046361 0.82 AHR (0.62) AHRALDH1A1NR4A2TRPA1CA1
Quinoline SCHEMBL28826923 0.82 NR4A2 (0.63) AHRALDH1A1METAP2METAP1CBFB
Quinoline SCHEMBL27735425 0.82 ALDH1A1 (0.54) AHRALDH1A1METAP2NR4A2TRPA1
Quinoline SCHEMBL27740778 0.81 NPC1 (0.51) AHRALDH1A1NR4A2TRPA1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108368106-A FUSED HETEROCYCLIC COMPOUND DERIVATIVE AND APPLICATION THEREOF 江苏恩华药业股份有限公司 2018-08-03 CN disclosed
CN-106608875-A Synthesis and application of fused heterocycle derivative 江苏恩华药业股份有限公司 2017-05-03 CN disclosed
CN-105814019-A Urea derivative or pharmacologically acceptable salt thereof 杏林制药株式会社 2016-07-27 CN disclosed
CN-105367474-A Indoline derivative and application of indoline derivative in medicine GUANGDONG HEC PHARMACEUTICAL 2016-03-02 CN disclosed
CN-102066326-A Pyridone compound ASTELLAS PHARMA INC 2011-05-18 CN disclosed
CN-101233132-A Compounds for modulating TRPV3 function HYDRA BIOSCIENCES INC (US) 2008-07-30 CN disclosed