Quinoline

Quinoline

SCHEMBL28046361

Brc1ccc2cc[nH]c2c1.c1ccc2ncccc2c1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 4/20 0.62
CYP1A2 P05177 1/20 0.58
CYP2C19 P33261 1/20 0.58
HTT P42858 1/20 0.58
ALDH1A1 P00352 3/20 0.50
NR4A2 P43354 2/20 0.45
CYP2A6 P11509 2/20 0.45
TRPA1 O75762 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
ITGB2 P05107 1/20 0.42
ICAM1 P05362 1/20 0.42
ITGAL P20701 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
ADK P55263 1/20 0.42
AXL P30530 1/20 0.41
NUDT1 P36639 1/20 0.41
EGFR P00533 1/20 0.41
MEN1 O00255 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27705544 0.88 AHR (0.62) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL843861 0.82 ALDH1A1 (0.63) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL28292512 0.82 ALDH1A1 (0.63) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL28816675 0.82 ALDH1A1 (0.63) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL28073739 0.82 ALDH1A1 (0.63) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL27735425 0.82 ALDH1A1 (0.54) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL27713201 0.82 AHR (0.62) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL28826923 0.82 NR4A2 (0.63) AHRCYP1A2CYP2C19HTTALDH1A1
Quinoline SCHEMBL27740778 0.81 NPC1 (0.51) AHRALDH1A1NR4A2TRPA1CA1
Quinoline SCHEMBL27739225 0.81 ALDH1A1 (0.61) AHRCYP1A2CYP2C19HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105769871-A Application of NIK protein kinase inhibitor in serving as medicine for treating liver diseases 东北师范大学 2016-07-20 CN disclosed
CN-105367474-A Indoline derivative and application of indoline derivative in medicine GUANGDONG HEC PHARMACEUTICAL 2016-03-02 CN disclosed
CN-105209457-A Pyrrolidine derivatives, pharmaceutical compositions containing them, and their use in therapy ABBVIE DEUTSCHLAND 2015-12-30 CN disclosed