SCHEMBL27714520

SCHEMBL27714520

Nc1ccccc1-c1cn2c[c]sc2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 5/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
NPC1 O15118 3/20 0.37
GAA P10253 3/20 0.37
RAB9A P51151 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MAPT P10636 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
AR P10275 1/20 0.36
IDO1 P14902 1/20 0.36
HSD17B10 Q99714 3/20 0.34
ATR Q13535 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
ADORA2A P29274 2/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL219596 0.75 TP53 (0.57) ALDH1A1SMN1; SMN2NPC1GAARAB9A
SCHEMBL13470761 0.71 TP53 (0.42) ALDH1A1KDM4ESMN1; SMN2NPC1GAA
SCHEMBL30714904 0.69 RAB9A (0.54) ALDH1A1KDM4ESMN1; SMN2NPC1GAA
SCHEMBL222164 0.69 RAB9A (0.54) ALDH1A1KDM4ESMN1; SMN2NPC1GAA
SCHEMBL218882 0.68 TP53 (0.43) ALDH1A1KDM4ESMN1; SMN2NPC1GAA
SCHEMBL27735301 0.66 NPC1 (0.38) ALDH1A1KDM4ESMN1; SMN2NPC1GAA
SCHEMBL218827 0.66 ALDH1A1 (0.62) ALDH1A1KDM4ESMN1; SMN2NPC1GAA
SCHEMBL11987212 0.64 SIRT1 (0.42) SMN1; SMN2MAPTARTP53
SCHEMBL18807101 0.64 SUV39H2 (0.46) ALDH1A1KDM4ESMN1; SMN2NPC1GAA
SCHEMBL4627970 0.64 RAB9A (0.51) ALDH1A1KDM4ESMN1; SMN2NPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101316853-B Benzothiazole and thiazolopyridine as SIRTUIN modulators SIRTRIS PHARMACEUTICALS INC 2014-09-24 CN disclosed
CN-103145738-A Imidazo [2,1-b] thiayole derivatives as SIRTUIN modulating compounds SIRTRIS PHARMACEUTICALS INC 2013-06-12 CN disclosed
CN-101316853-A Benzothiazole and thiazolopyridine as SIRTUIN modulators SIRTRIS PHARMACEUTICALS INC (US) 2008-12-03 CN disclosed
CN-101282761-A Benzimidazole derivatives as SIRTUIN modulators SIRTRIS PHARMACEUTICALS INC (US) 2008-10-08 CN disclosed
CN-101282974-A Benzimidazole derivatives as SIRTUIN modulators SIRTRIS PHARMACEUTICALS INC (US) 2008-10-08 CN disclosed
CN-101277963-A Benzimidazole derivatives as SIRTUIN modulators SIRTIS PHARMACEUTICALS INC (US) 2008-10-01 CN disclosed
CN-101277965-A Imidazo [2, 1-b ] thiazole derivatives as SIRTUIN modulating compounds SIRTRIS PHARMACEUTICALS INC (US) 2008-10-01 CN disclosed