Gliquidone

Gliquidone

SCHEMBL27714721

COc1ccc2c(c1)C(=O)N(CCc1ccc(S(=O)(=O)NC(=O)NC3CCCCC3)cc1)C(=O)C2(C)C.Cc1cc(C(=O)NCCc2ccc(S(=O)(=O)NC(=O)NC3CCCCC3)cc2)no1

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.78
LMNA P02545 4/20 0.78
CYP3A4 P08684 3/20 0.78
ABCC3 O15438 3/20 0.78
ABCC4 O15439 3/20 0.78
ABCB11 O95342 3/20 0.78
HIF1A Q16665 3/20 0.78
HTR2A P28223 2/20 0.78
TBXA2R P21731 2/20 0.78
NR1I3 Q14994 2/20 0.78
KDM4E B2RXH2 1/20 0.78
NR1I2 O75469 1/20 0.78
NR3C1 P04150 1/20 0.78
RARA P10276 1/20 0.78
RARB P10826 1/20 0.78
RARG P13631 1/20 0.78
HPGD P15428 1/20 0.78
NR1H2 P55055 1/20 0.78
PDE4D Q08499 1/20 0.78
NR1H3 Q13133 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gliquidone SCHEMBL21824303 0.91 CYP2C9 (0.79) CYP2C9LMNACYP3A4ABCC3ABCC4
Gliquidone SCHEMBL29465034 0.88 LMNA (1.00) CYP2C9LMNACYP3A4ABCC3ABCC4
Gliquidone SCHEMBL15669239 0.88 LMNA (1.00) CYP2C9LMNACYP3A4ABCC3ABCC4
Gliquidone SCHEMBL37769 0.88 LMNA (1.00) CYP2C9LMNACYP3A4ABCC3ABCC4
Gliquidone SCHEMBL676846 0.88 LMNA (0.98) CYP2C9LMNACYP3A4ABCC3ABCC4
Gliquidone SCHEMBL15845544 0.82 CYP2C9 (0.53) CYP2C9LMNACYP3A4ABCC3ABCC4
SCHEMBL8216020 0.82 LMNA (0.87) CYP2C9LMNACYP3A4ABCC3ABCC4
Gliquidone SCHEMBL28086518 0.81 LMNA (0.82) CYP2C9LMNACYP3A4ABCC3ABCC4
Glisolamide SCHEMBL38106 0.81 LMNA (0.73) CYP2C9LMNACYP3A4ABCC3ABCC4
Gliquidone SCHEMBL3112032 0.81 CYP2C9 (0.72) CYP2C9LMNACYP3A4ABCC3ABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101277960-A Acylated spiropiperidine derivatives as melanocortin-4 receptor modulators MERCK & CO INC (US) 2008-10-01 CN disclosed