Gliquidone

Gliquidone

SCHEMBL29465034

COc1ccc2c(c1)C(=O)N(CCc1ccc(S(=O)(=O)NC(=O)NC3CCCCC3)cc1)C(=O)C2(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 1.00
CYP3A4 P08684 4/20 1.00
CYP2C9 P11712 4/20 1.00
ABCC3 O15438 2/20 1.00
ABCC4 O15439 2/20 1.00
ABCB11 O95342 2/20 1.00
HTR2A P28223 2/20 1.00
HIF1A Q16665 2/20 1.00
HPGD P15428 2/20 1.00
KDM4E B2RXH2 1/20 1.00
NR1I2 O75469 1/20 1.00
NR3C1 P04150 1/20 1.00
RARA P10276 1/20 1.00
RARB P10826 1/20 1.00
RARG P13631 1/20 1.00
TBXA2R P21731 1/20 1.00
NR1H2 P55055 1/20 1.00
PDE4D Q08499 1/20 1.00
NR1H3 Q13133 1/20 1.00
PDE3A Q14432 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gliquidone SCHEMBL37769 1.00 LMNA (1.00) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL15669239 1.00 LMNA (1.00) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL676846 0.99 LMNA (0.98) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL8216020 0.93 LMNA (0.87) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL28086518 0.91 LMNA (0.82) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL21824303 0.89 CYP2C9 (0.79) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL27714721 0.88 CYP2C9 (0.78) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL10281162 0.86 CYP3A4 (0.76) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL11929012 0.86 CYP3A4 (0.76) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL25866045 0.86 CYP3A4 (0.75) LMNACYP3A4CYP2C9ABCC3ABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250376498-A1 FUSION PROTEINS COMPRISING AN IMPROVED GLP-1 RECEPTOR AGONIST AND USES THEREOF GUANGZHOU INNOGEN PHARMACEUTICAL GROUP CO LTD (CN) 2025-12-11 US claimed
EP-3758692-B1 COMPOSITIONS AND METHODS FOR TREATING PAIN UNIV MARYLAND (US) 2024-08-21 EP claimed
EP-4014999-B1 COMBINATION PRODUCT CONTAINING LIMONIN COMPOUND AND SULFONYLUREA DRUG ZHEJIANG YANGSHENGTANG INST OF NATURAL MEDICATION CO LTD (CN) 2023-11-29 EP claimed
EP-3359162-B1 METHODS OF TREATING INJURIES OR CONDITIONS RELATED TO CNS EDEMA BIOGEN CHESAPEAKE LLC (US) 2022-12-21 EP claimed
EP-1931320-B1 MICROPARTICLES WITH MODIFIED RELEASE OF AT LEAST ONE ACTIVE PRINCIPLE AND ORAL DOSAGE FORM COMPRISING THE SAME FLAMEL IRELAND LTD (IE) 2022-06-15 EP claimed
EP-3411026-B1 USE OF STIMULATORS OF SOLUBLE GUANYLATE CYCLASE FOR THE TREATMENT OF NONALCOHOLIC STEATOHEPATITIS (NASH) CYCLERION THERAPEUTICS INC (US) 2022-03-09 EP claimed
US-20260076972-A1 ANTIDIABETIC MEDICATIONS BOEHRINGER INGELHEIM INT (DE) 2026-03-19 US disclosed
EP-4648849-A1 NMU RECEPTOR 2 AGONISTS Boehringer Ingelheim International GmbH (DE) 2025-11-19 EP disclosed
US-20250312456-A1 TREATMENT FOR DIABETES IN PATIENTS INAPPROPRIATE FOR METFORMIN THERAPY BOEHRINGER INGELHEIM INT (DE) 2025-10-09 US disclosed
US-12364700-B2 Medical use of pharmaceutical combination or composition BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2025-07-22 US disclosed
US-12312352-B2 Use of a DPP-4 inhibitor in SIRS and/or sepsis BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2025-05-27 US disclosed
EP-4031108-B1 EXTRUDED DEPOT FORM FOR CONTROLLED ACTIVE SUBSTANCE RELEASE AMW GMBH (DE) 2025-04-02 EP disclosed
US-20250082642-A1 TREATMENT FOR DIABETES IN PATIENTS WITH INSUFFICIENT GLYCEMIC CONTROL DESPITE THERAPY WITH AN ORAL OR NON-ORAL ANTIDIABETIC DRUG BOEHRINGER INGELHEIM INT (DE) 2025-03-13 US disclosed
EP-2849754-B1 LINAGLIPTIN, A XANTHINE DERIVATIVE AS DPP-4 INHIBITOR, FOR USE IN THE TREATMENT OF SIRS AND/OR SEPSIS BOEHRINGER INGELHEIM INT (DE) 2022-09-14 EP disclosed
EP-2397142-B1 Use of DPP IV inhibitors BOEHRINGER INGELHEIM INT (DE) 2022-07-27 EP disclosed
US-11369645-B2 Hafnia alvei impact on regulation of appetite and metabolic syndrome aspects INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-28 US disclosed
US-20220184088-A1 USES OF DPP IV INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2022-06-16 US disclosed
US-20220160717-A1 Cardio- and Renosafe Antidiabetic Therapy BOEHRINGER INGELHEIM INT (DE) 2022-05-26 US disclosed
US-11291668-B2 Uses of DPP IV inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-04-05 US disclosed
US-20220088023-A1 ANTIDIABETIC MEDICATIONS BOEHRINGER INGELHEIM INT (DE) 2022-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250376498-A1 FUSION PROTEINS COMPRISING AN IMPROVED GLP-1 RECEPTOR AGONIST AND USES THEREOF GLP1R, GIPR, GCGR LMNA 4415/4885CYP3A4 4606/4885CYP2C9 4524/4885
US-20220184088-A1 USES OF DPP IV INHIBITORS DPP4, DPP3, DPP7 LMNA 3770/4885CYP3A4 175/4885CYP2C9 627/4885
US-20250082642-A1 TREATMENT FOR DIABETES IN PATIENTS WITH INSUFFICIENT GLYCEMIC CONTROL DESPITE THERAPY WITH AN ORAL OR NON-ORAL ANTIDIABETIC DRUG DPP4, DPP3, DPP7 LMNA 4808/4885CYP3A4 129/4885CYP2C9 825/4885
US-20220088023-A1 ANTIDIABETIC MEDICATIONS SLC5A1, SLC5A2, DPP4 LMNA 3799/4885CYP3A4 599/4885CYP2C9 1458/4885
US-11291668-B2 Uses of DPP IV inhibitors DPP4, DPP3, DPP7 LMNA 3770/4885CYP3A4 175/4885CYP2C9 627/4885
US-20250312456-A1 TREATMENT FOR DIABETES IN PATIENTS INAPPROPRIATE FOR METFORMIN THERAPY DPP4, DPP3, DPP7 LMNA 4606/4885CYP3A4 78/4885CYP2C9 376/4885
US-12312352-B2 Use of a DPP-4 inhibitor in SIRS and/or sepsis DPP4, DPP3, DPP7 LMNA 4617/4885CYP3A4 147/4885CYP2C9 1106/4885
US-20260076972-A1 ANTIDIABETIC MEDICATIONS IAPP, DPP4, PYGL LMNA 1252/4885CYP3A4 1702/4885CYP2C9 3700/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.