Gliquidone

Gliquidone

SCHEMBL37769

COc1ccc2c(c1)C(=O)N(CCc1ccc(S(=O)(=O)NC(=O)NC3CCCCC3)cc1)C(=O)C2(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 1.00
CYP3A4 P08684 4/20 1.00
CYP2C9 P11712 4/20 1.00
ABCC3 O15438 2/20 1.00
ABCC4 O15439 2/20 1.00
ABCB11 O95342 2/20 1.00
HTR2A P28223 2/20 1.00
HIF1A Q16665 2/20 1.00
HPGD P15428 2/20 1.00
KDM4E B2RXH2 1/20 1.00
NR1I2 O75469 1/20 1.00
NR3C1 P04150 1/20 1.00
RARA P10276 1/20 1.00
RARB P10826 1/20 1.00
RARG P13631 1/20 1.00
TBXA2R P21731 1/20 1.00
NR1H2 P55055 1/20 1.00
PDE4D Q08499 1/20 1.00
NR1H3 Q13133 1/20 1.00
PDE3A Q14432 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gliquidone SCHEMBL15669239 1.00 LMNA (1.00) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL29465034 1.00 LMNA (1.00) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL676846 0.99 LMNA (0.98) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL8216020 0.93 LMNA (0.87) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL28086518 0.91 LMNA (0.82) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL21824303 0.89 CYP2C9 (0.79) LMNACYP3A4CYP2C9ABCC3ABCC4
Gliquidone SCHEMBL27714721 0.88 CYP2C9 (0.78) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL10281162 0.86 CYP3A4 (0.76) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL11929012 0.86 CYP3A4 (0.76) LMNACYP3A4CYP2C9ABCC3ABCC4
SCHEMBL25866045 0.86 CYP3A4 (0.75) LMNACYP3A4CYP2C9ABCC3ABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10493 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260124282-A1 DECORIN FOR ITS USE IN THE TREATMENT OF DIABETES CENTRE EUROPEEN D'ETUDE DU DIABETE (FR) 2026-05-07 US claimed
US-20260115210-A1 METHOD FOR TREATING SUBJECTS SUFFERING FROM CENTRAL NERVOUS SYSTEM CONTUSIONS REMEDY PHARMACEUTICALS, INC. (US) 2026-04-30 US claimed
US-12611416-B2 Methods of treating ischemic stroke at risk for cerebral or cerebellar edema REMEDY PHARMACEUTICALS, INC. (US) 2026-04-28 US claimed
EP-4714927-A1 A REACTIVE RESIN COMPOSITION COMPRISING A PEROXIDE-FREE INITIATOR SYSTEM WITH A SULFINATE AND A TERTIARY AMINE Hilti Aktiengesellschaft (LI) 2026-03-25 EP claimed
EP-4714925-A1 A REACTIVE RESIN COMPOSITION COMPRISING A PEROXIDE-FREE INITIATOR SYSTEM Hilti Aktiengesellschaft (LI) 2026-03-25 EP claimed
EP-4714928-A1 A REACTIVE RESIN COMPOSITION COMPRISING A PEROXIDE-FREE INITIATOR SYSTEM WITH A HETEROCYCLIC COMPOUND COMPRISING AT LEAST ONE N-N SINGLE BOND Hilti Aktiengesellschaft (LI) 2026-03-25 EP claimed
EP-4714926-A1 A REACTIVE RESIN COMPOSITION COMPRISING A PEROXIDE-FREE INITIATOR SYSTEM WITH A TERTIARY AMINE Hilti Aktiengesellschaft (LI) 2026-03-25 EP claimed
EP-4691496-A1 PHARMACEUTICAL PREPARATION CONTAINING GLP-1 FUSION PROTEIN AND USE THEREOF Guangzhou Innogen Pharmaceutical Group Co., Ltd. (CN) 2026-02-11 EP claimed
EP-4684799-A2 ANTIBODIES THAT DISRUPT THE INTERACTION OF GAL3 AND INSULIN RECEPTOR OR INTEGRINS AND METHODS OF USE THEREOF TrueBinding, Inc. (US) 2026-01-28 EP claimed
EP-4680240-A1 METHOD OF TREATING DISORDERS WITH SURF1 MALFUNCTION Cure Mito Foundation (US) 2026-01-21 EP claimed
US-5859037-A MIXTURE SYNERGISTIC FOR THE TREATMENT OF NON-INSULIN DEPENDENT DIABETES MELLITUS IN HUMANS, WHICH ALSO IMPROVES GLYCEMIC CONTROL WARNER-LAMBERT COMPANY (US) 1999-01-12 US claimed
WO-1998056378-A1 NOVEL NIDDM REGIMEN NOVO NORDISK A/S (DK) 1998-12-17 WO claimed
CN-1195531-A Drug for curing diabetes and its preparing method YAO YUANLIN (CN) 1998-10-14 CN claimed
WO-1998036755-A1 SULFONYLUREA-GLITAZONE SYNERGISTIC COMBINATIONS FOR DIABETES WARNER LAMBERT COMPANY (US) 1998-08-27 WO claimed
WO-1997041857-A1 COMPOSITION COMPRISING A KATP CHANNEL INHIBITOR FOR USE IN THE TREATMENT OF HEMORRHAGIC SHOCK CHILDREN'S HOSPITAL MEDICAL CENTER (US) 1997-11-13 WO claimed
CN-1156403-A Highly active sulphonyl urea preparations exhibiting rapid or controlled release of the active substance, and method of producing them BRITISH TECHNOLOGY GROUP CO LT (GB) 1997-08-06 CN claimed
EP-0128483-B1 GALENIC FORMS OF ORAL ANTIDIABETICS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP claimed
EP-0128482-B1 GALENIC FORMS OF ORAL ANTIDIABETICS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-01-31 EP claimed
US-4708868-A Oral anti-diabetic pharmaceutical forms and the preparation thereof DR. KARL THOMAE GMBH (DE) 1987-11-24 US claimed
US-4696815-A Anti-diabetic pharmaceutical forms and the preparation thereof DR. KARL THOMAE GMBH (DE) 1987-09-29 US claimed