SCHEMBL2771809

SCHEMBL2771809

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1CCOc1cc2ccccc2cc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.54
MAPK14 Q16539 2/20 0.39
PPARG P37231 4/20 0.37
PPARA Q07869 4/20 0.37
MCL1 Q07820 4/20 0.35
BCL2 P10415 3/20 0.35
PPARD Q03181 2/20 0.35
FFAR1 O14842 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.34
NR1I2 O75469 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2771389 0.93 NR1H4 (0.54) NR1H4MAPK14PPARGPPARAMCL1
SCHEMBL2772157 0.92 NR1H4 (0.53) NR1H4MAPK14PPARGPPARAPPARD
SCHEMBL2773708 0.92 NR1H4 (0.53) NR1H4MAPK14PPARGPPARAPPARD
SCHEMBL2786965 0.91 NR1H4 (0.52) NR1H4MAPK14PPARGPPARAPPARD
SCHEMBL2772849 0.88 NR1H4 (0.54) NR1H4MAPK14PPARGPPARAMCL1
SCHEMBL2772480 0.87 NR1H4 (0.60) NR1H4PPARGPPARAMRGPRX4
SCHEMBL2770890 0.87 NR1H4 (0.64) NR1H4PPARGPPARAMRGPRX4
SCHEMBL2787707 0.85 NR1H4 (0.59) NR1H4PPARDMRGPRX4
SCHEMBL2771269 0.83 NR1H4 (0.56) NR1H4PPARDFFAR1MRGPRX4
SCHEMBL2771151 0.83 NR1H4 (0.57) NR1H4MCL1BCL2PPARDMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed