SCHEMBL2773708

SCHEMBL2773708

Cc1ccc(OCCc2ccc(OCc3c(C(C)C)cnn3-c3c(Cl)cccc3Cl)cc2C)c(C(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 6/20 0.53
PPARG P37231 3/20 0.36
PPARA Q07869 3/20 0.36
MAPK14 Q16539 1/20 0.36
DHODH Q02127 2/20 0.35
PPARD Q03181 2/20 0.34
FFAR1 O14842 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2772157 0.94 NR1H4 (0.53) NR1H4PPARGPPARAMAPK14PPARD
SCHEMBL2786965 0.93 NR1H4 (0.52) NR1H4PPARGPPARAMAPK14PPARD
SCHEMBL2771389 0.92 NR1H4 (0.54) NR1H4PPARGPPARAMAPK14PPARD
SCHEMBL2771809 0.92 NR1H4 (0.54) NR1H4PPARGPPARAMAPK14PPARD
SCHEMBL2772849 0.88 NR1H4 (0.54) NR1H4PPARGPPARAMAPK14PPARD
SCHEMBL2772071 0.87 NR1H4 (0.56) NR1H4DHODHMRGPRX4
SCHEMBL2772480 0.87 NR1H4 (0.60) NR1H4PPARGPPARAMRGPRX4
SCHEMBL2770890 0.86 NR1H4 (0.64) NR1H4PPARGPPARAMRGPRX4
SCHEMBL2787707 0.85 NR1H4 (0.59) NR1H4PPARDMRGPRX4
SCHEMBL2773716 0.84 NR1H4 (0.52) NR1H4MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed