SCHEMBL27719795

SCHEMBL27719795

CNc1c(C)cc(N)cc1I

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
TSHR P16473 1/20 0.35
RAPGEF4 Q8WZA2 3/20 0.32
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14878894 0.84 ALDH1A1 (0.43) ALDH1A1TSHRRAPGEF4PDE10A
Hydrochloric Acid SCHEMBL10619129 0.81 ALDH1A1 (0.41) ALDH1A1TSHRRAPGEF4PDE10A
SCHEMBL27849756 0.77 CYP3A4 (0.41) ALDH1A1TSHR
SCHEMBL27725921 0.77
SCHEMBL27719791 0.74 CYP3A4 (0.45) ALDH1A1TSHRRAPGEF4
SCHEMBL27849706 0.72 GLA (0.38) TSHR
SCHEMBL20344365 0.70 TTR (0.48) ALDH1A1TSHRPDE10A
SCHEMBL13928793 0.68 ALDH1A1 (0.38) ALDH1A1TSHRPDE10A
SCHEMBL526416 0.68 ALDH1A1 (0.47) ALDH1A1TSHRPDE10A
SCHEMBL112391 0.67 ALDH1A1 (0.53) ALDH1A1TSHRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101142174-B Novel compound as vanilloid receptor antagonist, isomer thereof or pharmaceutically acceptable salt thereof, and pharmaceutical composition comprising the same AMOREPACIFIC CORP 2012-05-09 CN disclosed
CN-101163670-A Novel compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist, and pharmaceutical compositions containing the same AMOREPACIFIC CORP (KR) 2008-04-16 CN disclosed
CN-101142174-A Novel compounds as vanilloid receptor antagonists, isomers thereof or pharmaceutically acceptable salts thereof; and pharmaceutical compositions comprising the same AMOREPACIFIC CORP (KR) 2008-03-12 CN disclosed