SCHEMBL27720173

SCHEMBL27720173

[CH2]CCc1csc(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 8/20 0.56
MAPT P10636 4/20 0.56
KDM4E B2RXH2 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
TP53 P04637 14/20 0.55
POLB P06746 2/20 0.54
HTT P42858 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3370362 0.86 LMNA (0.58) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL27912402 0.86 LMNA (0.55) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL4905756 0.86 LMNA (0.55) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL6343767 0.86 LMNA (0.55) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL4903824 0.84 LMNA (0.53) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL4907133 0.84 LMNA (0.56) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL12151145 0.83 POLB (0.55) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL2236881 0.83 GFER (0.66) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL7895624 0.83 LMNA (0.51) LMNAMAPTKDM4ESMN1; SMN2TP53
SCHEMBL4553327 0.83 LMNA (0.51) LMNAMAPTKDM4ESMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101287718-A Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER PROD INC (US) 2008-10-15 CN disclosed