SCHEMBL27720378

SCHEMBL27720378

Cc1ncc(NC(=O)c2cc(F)cc(C(F)(F)F)c2)cc1NC(=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.55
CSF1R P07333 3/20 0.54
KIT P10721 2/20 0.54
P2RX1 P51575 1/20 0.52
AURKA O14965 1/20 0.48
BRAF P15056 6/20 0.48
KCNK3 O14649 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
NR2E1 Q9Y466 1/20 0.48
VNN1 O95497 1/20 0.47
KCNQ3 O43525 1/20 0.47
KCNQ2 O43526 1/20 0.47
KCNE1 P15382 1/20 0.47
KCNQ1 P51787 1/20 0.47
KCNQ5 Q9NR82 1/20 0.47
LMNA P02545 1/20 0.47
RAF1 P04049 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27699760 0.87 KCNQ3 (0.53) PIK3CACSF1RP2RX1AURKABRAF
SCHEMBL27720393 0.84 MEN1 (0.61) KCNK3NPC1RAB9AKCNQ3KCNQ2
SCHEMBL27699924 0.83 LCK (0.60) CSF1RKITBRAF
Cyclopropane SCHEMBL27720374 0.81 MEN1 (0.57) CSF1RKITKCNK3NPC1RAB9A
SCHEMBL27720423 0.81 KCNQ3 (0.58) CSF1RKITBRAFNPC1RAB9A
SCHEMBL27720418 0.80 CSF1R (0.50) CSF1RKITBRAFNPC1RAB9A
SCHEMBL27699900 0.78 BRAF (0.52) CSF1RKITBRAFRAB9AKCNQ3
SCHEMBL27720500 0.77 KMT2A (0.64) KCNK3NPC1RAB9A
SCHEMBL7745683 0.76 P2RX1 (0.82) P2RX1KCNK3NPC1RAB9ANR2E1
SCHEMBL28772278 0.75 KCNQ3 (0.62) KCNK3NPC1RAB9AKCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128454-A Pyridine carboxamide derivatives for use as anticancer agents ASTRAZENECA AB (SE) 2008-02-20 CN disclosed