SCHEMBL27722652

SCHEMBL27722652

CCCC(C=O)c1ccccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 1/20 0.39
HSD11B1 P28845 3/20 0.39
CNR2 P34972 2/20 0.38
CTSS P25774 4/20 0.37
MC4R P32245 1/20 0.37
CTSK P43235 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
TSHR P16473 2/20 0.36
CYP2C19 P33261 2/20 0.36
MAPK1 P28482 2/20 0.35
POLB P06746 1/20 0.35
SLC6A4 P31645 1/20 0.35
P2RX7 Q99572 1/20 0.35
EPHX2 P34913 1/20 0.34
PPARG P37231 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27626781 0.80 ACP3 (0.41) ACP3HSD11B1CNR2CTSSMC4R
SCHEMBL27742156 0.78 ACP3 (0.37) ACP3HSD11B1CNR2CTSSMC4R
SCHEMBL5609116 0.78 ACP3 (0.41) ACP3HSD11B1CNR2MC4RCYP1A2
SCHEMBL27925756 0.78 TAS1R3 (0.39) CNR2MC4RCYP3A4CYP2C9MAPT
SCHEMBL19879071 0.78 MC4R (0.41) ACP3HSD11B1CNR2MC4RCYP1A2
SCHEMBL27907690 0.77 KCNK3 (0.37) TSHRSLC6A4EPHX2PPARG
SCHEMBL16442475 0.76 P2RX7 (0.42) ACP3HSD11B1CNR2MC4RCYP1A2
SCHEMBL21311456 0.76 P2RX7 (0.42) ACP3HSD11B1CNR2MC4RCYP1A2
SCHEMBL12944872 0.76 MC4R (0.40) ACP3HSD11B1CNR2MC4RCYP1A2
SCHEMBL1824153 0.76 ESR1 (0.39) ACP3MC4RCYP3A4CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101326155-B Propionamide compounds as antiinflammatory agents HOFFMANN LA ROCHE 2012-06-20 CN disclosed
CN-101326169-B Glucocorticoid receptor modulators as antiinflammatory agents HOFFMANN LA ROCHE 2011-11-16 CN disclosed
CN-101326155-A Propionamide compounds as antiinflammatory agents HOFFMANN LA ROCHE (CH) 2008-12-17 CN disclosed
CN-101326169-A Glucocorticoid receptor modulators as antiinflammatory agents HOFFMANN LA ROCHE (CH) 2008-12-17 CN disclosed