SCHEMBL27723969

SCHEMBL27723969

CCc1c(N)cc(Cl)c(CC)c1NC(=O)N(CCc1ccc(OC(F)(F)F)cc1)c1ccc(C(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 2/20 0.36
GCGR P47871 3/20 0.35
GIPR P48546 2/20 0.35
TRPV1 Q8NER1 2/20 0.34
EPHX1 P07099 1/20 0.34
NPBWR1 P48145 1/20 0.34
MCHR1 Q99705 1/20 0.34
GLP1R P43220 1/20 0.34
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
CACNA1G O43497 1/20 0.32
CACNA1H O95180 1/20 0.32
CACNA1I Q9P0X4 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
KMT2A Q03164 1/20 0.32
PPARG P37231 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591412 0.92 GCGR (0.42) ALDH1A1CYP3A4GCGRGIPRNPBWR1
SCHEMBL27724115 0.91 CYP3A4 (0.35) ALDH1A1CYP3A4NPC1PPARGPPARD
SCHEMBL27703384 0.89 UTS2R (0.40) MCHR1PDK1
SCHEMBL27703386 0.88 CYP3A4 (0.38) ALDH1A1CYP3A4MEN1KMT2A
SCHEMBL4592518 0.87 CYP3A4 (0.34) CYP3A4CACNA1HNR1H4
SCHEMBL27703387 0.86 RAB9A (0.39) ALDH1A1CYP3A4EPHX1MEN1NPC1
SCHEMBL27724006 0.84 PSMB5 (0.35) ALDH1A1CYP3A4GLP1R
SCHEMBL27703435 0.82 CHRM5 (0.36) ALDH1A1CYP3A4MEN1KMT2APDK1
SCHEMBL27723968 0.82 EPHX2 (0.37) ALDH1A1CYP3A4MEN1KMT2A
SCHEMBL4592219 0.81 MAPT (0.37) ALDH1A1CYP3A4NPC1NLRP3NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101189209-A C5a receptor antagonists JERINI AG (DE) 2008-05-28 CN claimed
CN-101189209-A C5a receptor antagonists JERINI AG (DE) 2008-05-28 CN disclosed