SCHEMBL27724006

SCHEMBL27724006

CCc1c(N)cc(Cl)c(CC)c1NC(=O)N(CCc1ccc(S(C)(=O)=O)cc1)c1ccc(C(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.35
RORC P51449 1/20 0.34
MAPK8 P45983 2/20 0.33
MAPK9 P45984 2/20 0.33
MAPK10 P53779 2/20 0.33
CNR2 P34972 2/20 0.33
CYP3A4 P08684 1/20 0.33
ALDH1A1 P00352 1/20 0.32
F10 P00742 4/20 0.32
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
PRKD3 O94806 1/20 0.32
MAPK1 P28482 1/20 0.32
PRKD2 Q9BZL6 1/20 0.32
BMP1 P13497 1/20 0.32
GLP1R P43220 1/20 0.32
EGFR P00533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591584 0.91 CNR2 (0.37) RORCMAPK8MAPK9MAPK10CNR2
SCHEMBL27724115 0.91 CYP3A4 (0.35) CYP3A4ALDH1A1F10PRSS1PRSS2
SCHEMBL27703386 0.90 CYP3A4 (0.38) CNR2CYP3A4ALDH1A1TP53MAPT
SCHEMBL4592518 0.89 CYP3A4 (0.34) CNR2CYP3A4F10TP53MAPT
SCHEMBL27703387 0.88 RAB9A (0.39) CNR2CYP3A4ALDH1A1MAPTEGFR
SCHEMBL27703384 0.86 UTS2R (0.40) PSMB5RORCTP53MAPTEGFR
SCHEMBL27723969 0.84 ALDH1A1 (0.39) CYP3A4ALDH1A1GLP1R
SCHEMBL27723968 0.82 EPHX2 (0.37) CNR2CYP3A4ALDH1A1MAPT
SCHEMBL4592219 0.82 MAPT (0.37) CNR2CYP3A4ALDH1A1TP53MAPT
SCHEMBL27723970 0.82 TAAR1 (0.36) CNR2CYP3A4TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101189209-A C5a receptor antagonists JERINI AG (DE) 2008-05-28 CN disclosed