SCHEMBL27724973

SCHEMBL27724973

O=C(O)c1n[c]sc1NC1CC1

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 3/20 0.37
CSNK2A1 P68400 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2830009 0.71 HCAR3 (0.44) HCAR3CSNK2A1
SCHEMBL3580737 0.70 HCAR3 (0.42) HCAR3CSNK2A1
SCHEMBL3584391 0.67 ALDH1A1 (0.37) HCAR3
SCHEMBL2827434 0.66 HCAR3 (0.46) HCAR3
SCHEMBL2827656 0.65 HCAR3 (0.45) HCAR3
SCHEMBL8628930 0.62
SCHEMBL2443626 0.59 LDHA (0.30)
SCHEMBL9203287 0.59 HCAR3 (0.35) HCAR3
Lithium Ion SCHEMBL3580735 0.59 HCAR3 (0.35) HCAR3CSNK2A1
SCHEMBL8553614 0.59 ALDH1A1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101137653-B Thiazole-4-carboxamide derivatives as MGLUR5 antagonists HOFFMANN LA ROCHE 2012-05-09 CN claimed
CN-101137653-A Thiazole-4-carboxamide derivatives as MGLUR5 antagonists HOFFMANN LA ROCHE (CH) 2008-03-05 CN claimed
CN-101137653-B Thiazole-4-carboxamide derivatives as MGLUR5 antagonists HOFFMANN LA ROCHE 2012-05-09 CN disclosed
CN-101379036-B Anthranilamide/2-amino-heteroarene carboxamide derivatives HOFFMANN LA ROCHE 2011-06-01 CN disclosed
CN-101379036-A Anthranilamide/2-amino-heteroarene carboxamide derivatives HOFFMANN LA ROCHE (CH) 2009-03-04 CN disclosed
CN-101137653-A Thiazole-4-carboxamide derivatives as MGLUR5 antagonists HOFFMANN LA ROCHE (CH) 2008-03-05 CN disclosed