SCHEMBL27730489

SCHEMBL27730489

CN(C(=O)C1CCN(OC(=O)C(C)(C)C)CC1)c1ccc(F)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 8/20 0.43
MLNR O43193 3/20 0.35
EPHX2 P34913 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
F10 P00742 1/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
USP30 Q70CQ3 1/20 0.32
CYP46A1 Q9Y6A2 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27709993 0.87 PDK2 (0.52) PDK2EPHX2TDP1CYP46A1POLB
SCHEMBL27730506 0.85 PDK2 (0.38) PDK2SMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL27730541 0.84 POLB (0.37) PDK2SMN1; SMN2USP30POLB
SCHEMBL3182755 0.84 PDK2 (0.47) PDK2SMN1; SMN2KMT2AMEN1USP30
SCHEMBL27710057 0.77 TP53 (0.55) EPHX2SMN1; SMN2KMT2AMEN1POLB
SCHEMBL27805795 0.75 GPR119 (0.41) SMN1; SMN2
SCHEMBL27621448 0.73 MAPT (0.38) SMN1; SMN2ALDH1A1
SCHEMBL4875392 0.73 USP30 (0.47) EPHX2ALDH1A1KMT2AMEN1USP30
SCHEMBL27771460 0.73 SCD (0.49)
SCHEMBL28264100 0.72 PDK2 (0.60) PDK2MLNRSMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101227903-A Novel 3-spirocyclic indolyl derivatives as ORL-1 receptor modulators JANSSEN PHARMACEUTICA NV (BE) 2008-07-23 CN disclosed