SCHEMBL27735562

SCHEMBL27735562

CC(C)c1nc(CCNC(=O)OC(C)(C)C)no1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 3/20 0.41
GFER P55789 1/20 0.41
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
NQO2 P16083 1/20 0.39
CYP1A2 P05177 1/20 0.38
CTSK P43235 1/20 0.38
PCSK9 Q8NBP7 1/20 0.38
MAPT P10636 1/20 0.37
LMNA P02545 2/20 0.36
BCHE P06276 1/20 0.36
STK17B O94768 1/20 0.36
STK17A Q9UEE5 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24387803 0.83 HTT (0.51) HTTNPSR1ALDH1A1GFERGAA
SCHEMBL2830746 0.80 RAB9A (0.38) HTTALDH1A1LMNA
SCHEMBL27714548 0.79 BMP1 (0.35) HTTALDH1A1KMT2ALMNA
SCHEMBL13188592 0.78 HTT (0.43) HTTNPSR1ALDH1A1GFERGAA
SCHEMBL3718792 0.77 HTT (0.43) HTTNPSR1ALDH1A1GFERGAA
SCHEMBL1785524 0.76 HTT (0.50) HTTNPSR1ALDH1A1GFERGAA
SCHEMBL4213195 0.76 HTT (0.50) HTTNPSR1ALDH1A1GFERGAA
SCHEMBL3951349 0.75 HTT (0.51) HTTNPSR1ALDH1A1GFERGAA
SCHEMBL4223857 0.75 HTT (0.64) HTTNPSR1ALDH1A1GAAMEN1
SCHEMBL19384814 0.74 HTT (0.48) HTTNPSR1ALDH1A1GFERGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101248054-B Thiazole derivatives and use thereof MERCK SERONO SA 2012-05-09 CN disclosed
CN-101248054-A Thiazole derivatives and use thereof SERONO LAB (CH) 2008-08-20 CN disclosed