SCHEMBL27736210

SCHEMBL27736210

O=CC(=O)C1CCCNC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 4/20 0.61
SLC6A11 P48066 3/20 0.61
SLC6A13 Q9NSD5 3/20 0.61
TSHR P16473 2/20 0.61
LMNA P02545 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
KMT2A Q03164 2/20 0.59
KDM4E B2RXH2 1/20 0.59
MAPT P10636 1/20 0.59
ATM Q13315 1/20 0.59
CYP2D6 P10635 1/20 0.59
NOS2 P35228 1/20 0.48
CPN1 P15169 2/20 0.40
CPB2 Q96IY4 2/20 0.40
GABRA5 P31644 3/20 0.35
GABRB2 P47870 3/20 0.35
APLNR P35414 2/20 0.35
SLC6A12 P48065 2/20 0.35
GABRA1 P14867 2/20 0.35
GABRA4 P48169 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27793461 0.87
SCHEMBL14206645 0.83 TSHR (0.46) SLC6A1SLC6A11SLC6A13TSHRLMNA
SCHEMBL28099042 0.83 TSHR (0.46) SLC6A1SLC6A11SLC6A13TSHRLMNA
SCHEMBL4772461 0.78 SLC6A1 (0.71) SLC6A1SLC6A11SLC6A13TSHRLMNA
Nipecotic Acid SCHEMBL456856 0.76 SLC6A1 (1.00) SLC6A1SLC6A11SLC6A13TSHRLMNA
(R)-Nipecotic Acid SCHEMBL29880539 0.76
(R)-Nipecotic Acid SCHEMBL520075 0.76
Nipecotic Acid SCHEMBL85677 0.76
(S)-Nipecotic Acid SCHEMBL254683 0.76
Hydrochloric Acid SCHEMBL27891040 0.76 SLC6A1 (0.68) SLC6A1SLC6A11SLC6A13TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109020874-A A kind of Eliquis intermediate and preparation method thereof 上海雅本化学有限公司 2018-12-18 CN claimed
CN-107108871-A The manufacture method of polyester 日本曹达株式会社 2017-08-29 CN claimed
CN-110016020-A Compound or pharmaceutically acceptable salt thereof, application and pharmaceutical composition thereof 铁木医药有限公司 2019-07-16 CN disclosed
CN-109384778-A Use of a compound or a pharmaceutically acceptable salt thereof for the manufacture of a medicament for the treatment of a disease, health condition or disorder 铁木医药有限公司 2019-02-26 CN disclosed
CN-109369635-A Compound or pharmaceutically acceptable salt thereof, application and pharmaceutical composition thereof 铁木医药有限公司 2019-02-22 CN disclosed
CN-108947985-A Compound and its preparation method and application as autophagy regulator 苏州偶领生物医药有限公司 2018-12-07 CN disclosed
CN-108912111-A compounds and pharmaceutical compositions 铁木医药有限公司 2018-11-30 CN disclosed
CN-105408328-B sGC stimulators 铁木医药有限公司 2018-11-16 CN disclosed
CN-106278968-B A kind of method for synthesizing sulfo-amino acid derivative 华东理工大学 2018-02-13 CN disclosed
CN-104817561-B The Piperidine inhibitors of JAK3 奥斯拜客斯制药有限公司 2017-06-13 CN disclosed
CN-106278968-A A kind of method synthesizing sulfo-amino acid derivative 华东理工大学 2017-01-04 CN disclosed
CN-105408328-A sGC stimulators IRONWOOD PHARMACEUTICALS INC 2016-03-16 CN disclosed
CN-104817561-A Piperidine inhibitors of Janus Kinase 3 AUSPEX PHARMACEUTICALS LLC 2015-08-05 CN disclosed
CN-102459270-B Piperidine inhibitors of janus kinase 3 AUSPEX PHARMACEUTICALS LLC 2015-04-29 CN disclosed
CN-103347873-A Pyrazole derivative and pest control agent NISSAN CHEMICAL IND LTD 2013-10-09 CN disclosed
CN-101243087-B 1,4-dihydropyridine-fused heterocycles, process for preparing the same, use and compositions containing them AVENTIS PHARMA SA 2013-07-24 CN disclosed
CN-101243087-A 1,4-dihydropyridine-fused heterocycles, process for preparing the same, use and compositions containing them AVENTIS PHARMA SA (FR) 2008-08-13 CN disclosed