SCHEMBL27736893

SCHEMBL27736893

c1ccc(-n2ccnc2C2CCCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICMT O60725 2/20 0.46
TNK2 Q07912 5/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
PKM P14618 1/20 0.40
MAPK1 P28482 1/20 0.39
FGFR2 P21802 1/20 0.39
HRH1 P35367 1/20 0.38
FDPS P14324 1/20 0.38
DRD1 P21728 1/20 0.37
DRD5 P21918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11264432 0.98 ICMT (0.45) ICMTTNK2NPC1RAB9ASMN1; SMN2
SCHEMBL13117192 0.85 ICMT (0.46) ICMTTNK2NPC1RAB9ASMN1; SMN2
SCHEMBL27736888 0.83 KCNH2 (0.48) ICMTTNK2MAPK1DRD1DRD5
SCHEMBL27736887 0.83 KDR (0.43) ICMTTNK2CYP1A2CYP3A4CYP2D6
SCHEMBL27837718 0.83 ICMT (0.40) ICMTTNK2FGFR2
SCHEMBL28779311 0.82 ICMT (0.41) ICMTTNK2
SCHEMBL25100064 0.79 TNK2 (0.41) ICMTTNK2NPC1RAB9ALMNA
SCHEMBL27736889 0.78 ICMT (0.49) ICMTRAB9AATM
SCHEMBL28019125 0.76 KCNH2 (0.55) ICMTCYP2D6
SCHEMBL28143054 0.76 ICMT (0.43) ICMTTNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101410114-B A3 adenosine receptor allosteric modulators US GOV HEALTH & HUMAN SERV (US) 2012-07-04 CN disclosed
CN-101410114-A A3 adenosine receptor allosteric modulators US GOV HEALTH & HUMAN SERV (US) 2009-04-15 CN disclosed