SCHEMBL27740964

SCHEMBL27740964

CCc1cc(CN(C)c2ccc(O)cc2F)ccc1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.36
CXCR3 P49682 1/20 0.36
EGFR P00533 2/20 0.36
LCK P06239 2/20 0.36
RARB P10826 2/20 0.36
RARA P10276 1/20 0.36
RARG P13631 1/20 0.36
ALDH1A1 P00352 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
TSHR P16473 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
HSD17B1 P14061 1/20 0.35
ESRRG P62508 1/20 0.35
PPARA Q07869 2/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27740953 0.88 EGFR (0.37) EGFRLCKRARBALDH1A1CA12
SCHEMBL27857292 0.85 NPC1 (0.39) CXCR3EGFRLCKALDH1A1CA12
SCHEMBL27761928 0.82 PPARA (0.41) CXCR3RARBRARARARGPPARA
SCHEMBL28780217 0.81 HSD17B1 (0.42) EGFRLCKALDH1A1CA12CA1
SCHEMBL497820 0.76 RXRA (0.41) EGFRLCKRARBALDH1A1CA12
SCHEMBL27762017 0.74 PLK1 (0.40) EGFRLCKALDH1A1ESRRGPPARA
SCHEMBL28126806 0.73 CA12 (0.57) EGFRLCKALDH1A1CA12CA1
SCHEMBL39010 0.73 CA12 (0.57) EGFRLCKALDH1A1CA12CA1
SCHEMBL3873135 0.72 CA12 (0.55) EGFRLCKALDH1A1CA12CA1
SCHEMBL27658957 0.72 CA12 (0.55) EGFRLCKALDH1A1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101448791-B Fxr agonists LILLY CO ELI 2011-11-16 CN disclosed
CN-101448798-A Compounds and methods for modulating FXR LILLY CO ELI (US) 2009-06-03 CN disclosed
CN-101448791-A FXR agonists LILLY CO ELI (US) 2009-06-03 CN disclosed