SCHEMBL27744679

SCHEMBL27744679

CC(C)(C)OC(=O)C1CC(Br)CN1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28044033 0.83 CHRM2 (0.33) MAPK1CHRM2CHRM1CHRM3
SCHEMBL4017978 0.80 DPP4 (0.41) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL21673908 0.80 DPP4 (0.41) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL31301933 0.80 CYP1A2 (0.42) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL695946 0.80 DPP4 (0.41) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL29308166 0.80 MAPK1 (0.36) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL12531141 0.80 MAPK1 (0.36) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL19901590 0.80 CYP1A2 (0.42) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL29308170 0.80 DPP4 (0.41) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL28146362 0.80 DPP4 (0.41) MAPK1L3MBTL1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101466726-B Azacyclo derivatives of androstanes and androstenes as medicaments for the treatment of cardiovascular disorders SIGMA TAU IND FARMACEUTI 2014-09-24 CN disclosed
CN-101466726-A Azacyclo derivatives of androstanes and androstenes as medicaments for the treatment of cardiovascular disorders SIGMA TAU IND FARMACEUTI (IT) 2009-06-24 CN disclosed