SCHEMBL27744909

SCHEMBL27744909

Nc1onc(C(F)(F)F)c1-c1ccncc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 9/20 0.61
MAPK14 Q16539 2/20 0.54
KIF11 P52732 1/20 0.41
BRD4 O60885 2/20 0.40
MAPK9 P45984 1/20 0.39
MAPK10 P53779 1/20 0.39
MAPK11 Q15759 1/20 0.39
S1PR1 P21453 2/20 0.39
S1PR3 Q99500 2/20 0.39
TDO2 P48775 1/20 0.39
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SRC P12931 1/20 0.36
BRAF P15056 1/20 0.36
KDR P35968 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8764932 0.84 MLYCD (0.63) MLYCDBRD4TDO2
SCHEMBL10502800 0.83 MLYCD (0.66) MLYCDMAPK14BRD4MAPK9MAPK10
SCHEMBL10503592 0.81 MLYCD (0.64) MLYCDMAPK14BRD4TDO2
SCHEMBL10503952 0.81 MLYCD (0.64) MLYCDMAPK14BRD4TDO2
SCHEMBL10505666 0.78 MLYCD (0.59) MLYCDRAB9A
SCHEMBL4874434 0.76 MLYCD (1.00) MLYCD
SCHEMBL4327769 0.72 BRD4 (0.60) MLYCDMAPK14KIF11BRD4MAPK9
SCHEMBL4339786 0.71 MAPK14 (0.63) MLYCDMAPK14MAPK9MAPK10MAPK11
SCHEMBL8764291 0.71 BRD4 (0.53) MLYCDBRD4TDO2
SCHEMBL10731646 0.71 MLYCD (0.52) MLYCDBRD4NPC1RAB9ASRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101472921-B Pyridylisoxazole derivative ASKA PHARM CO LTD 2012-10-10 CN disclosed
CN-101472921-A Pyridylisoxazole derivative ASKA PHARM CO LTD (JP) 2009-07-01 CN disclosed